LT - MALEATE SALTS OF A B-RAF KINASE INHIBITOR, CRYSTALLINE FORMS, METHODS OF PREPARATION, AND USES THEREFORE
EN - MALEATE SALTS OF A B-RAF KINASE INHIBITOR, CRYSTALLINE FORMS, METHODS OF PREPARATION, AND USES THEREFORE
Legal status
Patent not validated
Bibliographic data
Indications of the International Patent Classification (IPC)
| (51) |
INT.CL. |
C07D 405/14 |
(2006.01) |
|
|
C07D 471/04 |
(2013.01) |
|
|
C07D 471/04 |
(2006.01) |
|
|
A61P 35/00 |
(2018.01) |
|
|
A61K 31/4184 |
(2006.01) |
|
|
A61K 31/4355 |
(2006.01) |
|
|
A61K 31/5585 |
(2006.01) |
|
|
A61P 35/00 |
(2006.01) |
European patent
| (11) |
Number of the document |
3283486 |
| (13) |
Kind of document |
T |
| (96) |
European patent application number |
16779601.0 |
|
Date of filing the European patent application |
2016-04-14 |
| (97) |
Date of publication of the European application |
2018-02-21 |
| (45) |
Date of publication and mention of the grant of the patent |
2022-07-27
|
| (46) |
Date of publication of the claims translation |
|
PCT application
| (86) |
Number |
PCT/CN2016/079251 |
|
Date |
2016-04-14 |
PCT application publication
| (87) |
Number |
WO 2016/165626 |
|
Date |
2016-10-20 |
Priority applications
| (30) |
Number |
Date |
Country code |
|
PCT/CN2015/076639 |
2015-04-15
|
WO |
Inventors
| (72) |
ZHANG, Guoliang , CN
ZHOU, Changyou , US
|
Grantee
| (73) |
BeiGene, Ltd. ,
c/o Mourant Ozannes Corporate Services
(Cayman) Limited
94 Solaris Avenue, PO Box 1348
George Town, KY1-1108 Camana Bay, Grand Cayman,
KY
|
Title
| (54) |
MALEATE SALTS OF A B-RAF KINASE INHIBITOR, CRYSTALLINE FORMS, METHODS OF PREPARATION, AND USES THEREFORE |
| |
MALEATE SALTS OF A B-RAF KINASE INHIBITOR, CRYSTALLINE FORMS, METHODS OF PREPARATION, AND USES THEREFORE |