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LT - SELECTIVE ANDROGEN RECEPTOR DEGRADER (SARD) LIGANDS AND METHODS OF USE THEREOF
EN - SELECTIVE ANDROGEN RECEPTOR DEGRADER (SARD) LIGANDS AND METHODS OF USE THEREOF

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Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07C 271/02 (2006.01)
A61K 45/06 (2013.01)
A61K 45/06 (2006.01)
C07C 271/02 (2013.01)
A61K 31/325 (2006.01)
C07D 209/08 (2013.01)
C07D 215/18 (2013.01)
A61K 31/405 (2006.01)
A61P 35/00 (2006.01)
C07D 217/04 (2013.01)
C07D 209/42 (2006.01)
C07D 231/56 (2013.01)
C07D 235/16 (2006.01)
C07D 235/16 (2013.01)
C07D 487/04 (2006.01)
C07D 487/04 (2013.01)
C07D 209/42 (2013.01)
A61K 31/405 (2013.01)
A61K 31/416 (2013.01)
A61K 31/4184 (2013.01)
A61P 35/00 (2018.01)
A61K 31/403 (2013.01)
A61K 31/404 (2013.01)
European patent
(11) Number of the document 3286164
(13) Kind of document T
(96) European patent application number 16783866.3
Date of filing the European patent application 2016-04-21
(97) Date of publication of the European application 2018-02-28
(45) Date of publication and mention of the grant of the patent 2024-05-29
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2016/028674
Date 2016-04-21
PCT application publication
(87) Number WO 2016/172358
Date 2016-10-27
Priority applications
(30) Number Date Country code
201562150763 P 2015-04-21 US
201562220057 P 2015-09-17 US
201562220187 P 2015-09-17 US
201562219859 P 2015-09-17 US
201562241532 P 2015-10-14 US
Inventors
(72)
NARAYANAN, Ramesh , US
MILLER, Duane D. , US
PONNUSAMY, Thamarai , US
HWANG, Dong-Jin , US
HE, Yali , US
PAGADALA, Jayaprakash , US
DUKE, Charles B. , US
COSS, Christopher C. , US
DALTON, James T. , US
Grantee
(73) Oncternal Therapeutics, Inc. , 12230 El Camino Real Suite 230, San Diego CA 92130, US
University of Tennessee Research Foundation , 211 Conference Center Building 600 Henley Street, Knoxville, TN 37996, US
Title
(54) SELECTIVE ANDROGEN RECEPTOR DEGRADER (SARD) LIGANDS AND METHODS OF USE THEREOF
  SELECTIVE ANDROGEN RECEPTOR DEGRADER (SARD) LIGANDS AND METHODS OF USE THEREOF