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LT - ACYLATED 4-AMINOPIPERIDINES AS INHIBITORS OF SERINE PALMITOYLTRANSFERASE
EN - ACYLATED 4-AMINOPIPERIDINES AS INHIBITORS OF SERINE PALMITOYLTRANSFERASE

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 211/58 (2006.01)
A61K 31/437 (2006.01)
A61K 31/443 (2006.01)
A61K 31/4433 (2006.01)
A61K 31/4436 (2006.01)
A61K 31/4439 (2006.01)
A61K 31/444 (2006.01)
A61K 31/4468 (2006.01)
A61K 31/451 (2006.01)
A61K 31/452 (2006.01)
A61K 31/4709 (2006.01)
A61K 31/498 (2006.01)
A61K 31/506 (2006.01)
A61K 31/517 (2006.01)
A61K 31/5355 (2006.01)
A61K 31/661 (2006.01)
A61K 33/22 (2006.01)
A61P 35/00 (2006.01)
A61P 43/00 (2006.01)
C07D 215/42 (2006.01)
European patent
(11) Number of the document 3287441
(13) Kind of document T
(96) European patent application number 16783163.5
Date of filing the European patent application 2016-04-19
(97) Date of publication of the European application 2018-02-28
(45) Date of publication and mention of the grant of the patent 2021-06-09
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/JP2016/062418
Date 2016-04-19
PCT application publication
(87) Number WO 2016/171142
Date 2016-10-27
Priority applications
(30) Number Date Country code
2015086195 2015-04-20 JP
Inventors
(72)
ASANO, Yasutomi , JP
KOJIMA, Takuto , JP
KURASAWA, Osamu , JP
WONG, Tzu-Tshin , US
HIRATA, Yasuhiro , JP
IWAMURA, Naoki , JP
SAITO, Bunnai , JP
TANAKA, Yuta , JP
ARAI Ryosuke , JP
IMAMURA, Shinichi , JP
YONEMORI, Kazuko , JP
MIYAMOTO, Yasufumi , JP
KITAMURA, Shuji , JP
SANO, Osamu , JP
Grantee
(73) Takeda Pharmaceutical Company Limited , 1-1, Doshomachi 4-chome Chuo-ku, Osaka-shi, Osaka 541-0045, JP
Title
(54) ACYLATED 4-AMINOPIPERIDINES AS INHIBITORS OF SERINE PALMITOYLTRANSFERASE
  ACYLATED 4-AMINOPIPERIDINES AS INHIBITORS OF SERINE PALMITOYLTRANSFERASE