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LT - IMIDE-BASED MODULATORS OF PROTEOLYSIS AND ASSOCIATED METHODS OF USE
EN - IMIDE-BASED MODULATORS OF PROTEOLYSIS AND ASSOCIATED METHODS OF USE

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 401/14
C07D 495/14
A61P 35/00
European patent
(11) Number of the document 3302572
(13) Kind of document T
(96) European patent application number 16804586.2
Date of filing the European patent application 2016-06-03
(97) Date of publication of the European application 2018-04-11
(45) Date of publication and mention of the grant of the patent 2021-01-06
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2016/035874
Date 2016-06-03
PCT application publication
(87) Number WO 2016/197032
Date 2016-12-08
Priority applications
(30) Number Date Country code
201562171090 P 2015-06-04 US
201514792414 2015-07-06 US
Inventors
(72)
CREWS, Craig, M., US
CREW, Andrew, P., US
DONG, Hanqing, US
WANG, Jing, US
QIAN, Yimin, US
SIU, Kam, US
JIN, Meizhong, US
Grantee
(73) Arvinas Operations, Inc., 5 Science Park, New Haven, CT 06511, US
Title
(54) IMIDE-BASED MODULATORS OF PROTEOLYSIS AND ASSOCIATED METHODS OF USE
  IMIDE-BASED MODULATORS OF PROTEOLYSIS AND ASSOCIATED METHODS OF USE