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EN | LT
LT - CRYSTALLINE L-ARGININE SALT OF (R)-2-(7-(4-CYCLOPENTYL-3-(TRIFLUOROMETHYL)BENZYLOXY)-1,2,3,4-TETRAHYDROCYCLO-PENTA[B]INDOL-3-YL)ACETIC ACID FOR USE IN S1P1 RECEPTOR-ASSOCIATED DISORDERS
EN - CRYSTALLINE L-ARGININE SALT OF (R)-2-(7-(4-CYCLOPENTYL-3-(TRIFLUOROMETHYL)BENZYLOXY)-1,2,3,4-TETRAHYDROCYCLO-PENTA[B]INDOL-3-YL)ACETIC ACID FOR USE IN S1P1 RECEPTOR-ASSOCIATED DISORDERS

Teisinis statusas

Patentas neįsigaliojo (pagal EPK)

Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) INT.CL. C07D 209/94 (2006.01)
C07D 209/94 (2013.01)
A61K 31/403 (2006.01)
A61P 1/00 (2018.01)
A61P 37/00 (2006.01)
A61P 1/04 (2018.01)
A61P 29/00 (2006.01)
A61P 1/16 (2018.01)
A61P 35/00 (2006.01)
A61P 17/02 (2018.01)
A61P 17/06 (2018.01)
A61P 9/00 (2006.01)
A61P 1/00 (2006.01)
A61P 17/10 (2018.01)
A61P 7/00 (2006.01)
A61P 19/02 (2018.01)
A61P 3/00 (2006.01)
A61P 25/00 (2018.01)
A61P 29/00 (2018.01)
A61P 5/00 (2006.01)
A61P 3/00 (2018.01)
A61P 35/00 (2018.01)
A61P 37/00 (2018.01)
A61P 37/02 (2018.01)
A61P 43/00 (2018.01)
A61P 5/00 (2018.01)
A61P 7/00 (2018.01)
A61P 9/00 (2018.01)
A61P 3/10 (2018.01)
C07C 279/14 (2013.01)
Europos patentas
(11) Patento numeris 3310760
(13) Dokumento rūšis T
(96) Europos patento paraiškos numeris 16734529.7
Europos patento paraiškos padavimo data 2016-06-21
(97) Europos patento paraiškos paskelbimo data 2018-04-25
(45) Paskelbimo apie Europos patento išdavimą data 2022-09-14
(46) Apibrėžties vertimo paskelbimo data
Tarptautinės paraiškos padavimo
(86) Numeris PCT/US2016/038506
Data 2016-06-21
Tarptautinės paraiškos paskelbimo
(87) Numeris WO 2016/209809
Data 2016-12-29
Prioriteto paraiškos
(30) Numeris Data Šalis
201562182841 P 2015-06-22 US
201562207531 P 2015-08-20 US
Išradėjai
(72)
BLACKBURN, Anthony C. , US
CASTRO, Ryan O. , US
HADD, Mark A. , US
MA, You-An , US
MONTALBAN, Antonio Garrido , US
RUETER, Jaimie Karyn , US
SELVEY, Lee Alani , US
SHAKYA, Sagar Raj , US
CARLOS, Marlon , US
Savininkas
(73) Arena Pharmaceuticals, Inc. , 235 East 42nd Street, New York, NY 10017, US
Pavadinimas
(54) CRYSTALLINE L-ARGININE SALT OF (R)-2-(7-(4-CYCLOPENTYL-3-(TRIFLUOROMETHYL)BENZYLOXY)-1,2,3,4-TETRAHYDROCYCLO-PENTA[B]INDOL-3-YL)ACETIC ACID FOR USE IN S1P1 RECEPTOR-ASSOCIATED DISORDERS
  CRYSTALLINE L-ARGININE SALT OF (R)-2-(7-(4-CYCLOPENTYL-3-(TRIFLUOROMETHYL)BENZYLOXY)-1,2,3,4-TETRAHYDROCYCLO-PENTA[B]INDOL-3-YL)ACETIC ACID FOR USE IN S1P1 RECEPTOR-ASSOCIATED DISORDERS