|
|
Legal status
Patent not validated
| (51) | INT.CL. | C07D 403/12 | (2006.01) |
| C07D 403/12 | (2013.01) | ||
| C07D 413/14 | (2013.01) | ||
| C07D 413/14 | (2006.01) | ||
| C07D 401/10 | (2013.01) | ||
| C07D 401/10 | (2006.01) | ||
| C07D 407/14 | (2013.01) | ||
| C07D 403/10 | (2006.01) | ||
| C07D 413/10 | (2013.01) | ||
| C07D 403/14 | (2006.01) | ||
| C07D 417/10 | (2013.01) | ||
| C07D 407/14 | (2006.01) | ||
| C07D 417/14 | (2013.01) | ||
| C07D 413/10 | (2006.01) | ||
| C07D 417/10 | (2006.01) | ||
| C07D 471/04 | (2013.01) | ||
| C07D 417/14 | (2006.01) | ||
| C07D 403/10 | (2013.01) | ||
| C07D 471/04 | (2006.01) | ||
| C07D 403/14 | (2013.01) | ||
| A61P 31/04 | (2018.01) | ||
| A61K 31/41 | (2006.01) | ||
| A61K 31/4184 | (2006.01) | ||
| A61K 31/416 | (2013.01) | ||
| A61K 31/428 | (2006.01) | ||
| A61K 31/4184 | (2013.01) | ||
| A61K 31/4439 | (2006.01) | ||
| A61K 31/423 | (2013.01) | ||
| A61P 31/04 | (2006.01) | ||
| A61K 31/428 | (2013.01) | ||
| A61K 31/437 | (2013.01) | ||
| A61K 31/4375 | (2013.01) | ||
| A61K 31/4439 | (2013.01) | ||
| A61K 31/454 | (2013.01) | ||
| A61K 31/4545 | (2013.01) | ||
| A61K 31/4709 | (2013.01) | ||
| A61K 31/4725 | (2013.01) | ||
| A61K 31/498 | (2013.01) | ||
| A61K 31/5025 | (2013.01) | ||
| A61K 31/506 | (2013.01) | ||
| A61K 31/517 | (2013.01) | ||
| A61K 31/5377 | (2013.01) | ||
| C07D 401/14 | (2013.01) | ||
| C07D 487/04 | (2013.01) | ||
| A61K 31/198 | (2013.01) | ||
| A61K 31/407 | (2013.01) | ||
| A61K 31/41 | (2013.01) | ||
| A61K 31/4192 | (2013.01) | ||
| A61K 31/4196 | (2013.01) | ||
| A61K 31/421 | (2013.01) | ||
| A61K 31/4245 | (2013.01) | ||
| A61K 31/431 | (2013.01) | ||
| A61K 31/439 | (2013.01) | ||
| A61K 31/496 | (2013.01) | ||
| A61K 31/541 | (2013.01) | ||
| A61K 31/546 | (2013.01) | ||
| C07D 405/14 | (2013.01) | ||
| C07D 453/02 | (2013.01) | ||
| C07D 487/10 | (2013.01) | ||
| C07D 493/04 | (2013.01) | ||
| C07D 493/08 | (2013.01) | ||
| C07D 495/08 | (2013.01) |
| (11) | Number of the document | 3313828 |
| (13) | Kind of document | T |
| (96) | European patent application number | 16815358.3 |
| Date of filing the European patent application | 2016-06-24 | |
| (97) | Date of publication of the European application | 2018-05-02 |
| (45) | Date of publication and mention of the grant of the patent | 2023-07-12 |
| (46) | Date of publication of the claims translation |
| (86) | Number | PCT/US2016/039185 |
| Date | 2016-06-24 |
| (87) | Number | WO 2016/210234 |
| Date | 2016-12-29 |
| (30) | Number | Date | Country code |
| PCT/CN2015/082514 | 2015-06-26 | WO |
| (72) |
BENNETT, Frank , US
JIANG, Jinlong , US
PASTERNAK, Alexander , US
DONG, Shuzhi , US
GU, Xin , US
SCOTT, Jack, D. , US
TANG, Haiqun , US
ZHAO, Zhiqiang , US
HUANG, Yuhua , US
HUNTER, David , US
YANG, Dexi , US
YOUNG, Katherine , US
XIAO, Li , US
ZHANG, Zhibo , CN
FU, Jianmin , CN
BAI, Yunfeng , CN
ZHENG, Zhixiang , CN
ZHANG, Xu , CN
|
| (73) |
Merck Sharp & Dohme LLC ,
126 East Lincoln Avenue, Rahway, New Jersey 07065,
US
|
| (54) | METALLO-BETA-LACTAMASE INHIBITORS |
| METALLO-BETA-LACTAMASE INHIBITORS |