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LT - Kristalinė (S)-[3,4-difluoro-2-(2-fluoro-4-jodfenilamino)fenil] [3-hidroksi-3-(piperidin-2-IL) azetidin-1-IL]-metanono druska
EN - CRYSTALLINE FUMARATE SALT OF (S)-[3,4-DIFLUORO-2-(2-FLUORO-4-IODOPHENYLAMINO)PHENYL][3-HYDROXY-3-(PIPERIDIN-2-YL) AZETIDIN-1-YL]-METHANONE

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Patent in force

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 401/04 (2006.01)
A61K 31/397 (2006.01)
A61K 31/4427 (2006.01)
A61P 35/00 (2006.01)
European patent
(11) Number of the document 3317264
(13) Kind of document T
(96) European patent application number 16738971.7
Date of filing the European patent application 2016-06-30
(97) Date of publication of the European application 2018-05-09
(45) Date of publication and mention of the grant of the patent 2025-09-10
(46) Date of publication of the claims translation 2025-12-29
PCT application
(86) Number PCT/US2016/040444
Date 2016-06-30
PCT application publication
(87) Number WO 2017/004393
Date 2017-01-05
Priority applications
(30) Number Date Country code
201562187009 P 2015-06-30 US
Inventors
(72)
BROWN, Adrian St. Clair , GB
Grantee
(73) Exelixis, Inc. , 1851 Harbor Bay Parkway, Alameda, CA 94502, US
Attorney or representative
(74) Vitalija BANAITIENĖ, UAB TARPINĖ, A.P.Kavoliuko g. 24-152, LT-04328 Vilnius, LT
Title
(54) Kristalinė (S)-[3,4-difluoro-2-(2-fluoro-4-jodfenilamino)fenil] [3-hidroksi-3-(piperidin-2-IL) azetidin-1-IL]-metanono druska
  CRYSTALLINE FUMARATE SALT OF (S)-[3,4-DIFLUORO-2-(2-FLUORO-4-IODOPHENYLAMINO)PHENYL][3-HYDROXY-3-(PIPERIDIN-2-YL) AZETIDIN-1-YL]-METHANONE