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LT - CHIRAL DIARYL MACROCYCLES AS MODULATORS OF PROTEIN KINASES
EN - CHIRAL DIARYL MACROCYCLES AS MODULATORS OF PROTEIN KINASES

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 498/22
C07D 471/22
A61K 31/4985
A61K 31/519
European patent
(11) Number of the document 3317285
(13) Kind of document T
(96) European patent application number 16818768.0
Date of filing the European patent application 2016-06-30
(97) Date of publication of the European application 2018-05-09
(45) Date of publication and mention of the grant of the patent 2021-01-27
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2016/040329
Date 2016-06-30
PCT application publication
(87) Number WO 2017/004342
Date 2017-01-05
Priority applications
(30) Number Date Country code
201562188043 P 2015-07-02 US
201662353728 P 2016-06-23 US
Inventors
(72)
CUI, Jingrong J., US
LI, Yishan, US
ROGERS, Evan W., US
ZHAI, Dayong, US
DENG, Wei, US
UNG, Jane, US
Grantee
(73) Turning Point Therapeutics, Inc., 10628 Science Center Drive, Ste. 225, San Diego, CA 92121, US
Title
(54) CHIRAL DIARYL MACROCYCLES AS MODULATORS OF PROTEIN KINASES
  CHIRAL DIARYL MACROCYCLES AS MODULATORS OF PROTEIN KINASES