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LT - 5-(N-[6,5]-FUSED BICYCLIC ARYL TETRAHYDROISOQUINOLIN-6-YL) PYRIDIN-3-YL ACETIC ACID DERIVATIVES AS INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION
EN - 5-(N-[6,5]-FUSED BICYCLIC ARYL TETRAHYDROISOQUINOLIN-6-YL) PYRIDIN-3-YL ACETIC ACID DERIVATIVES AS INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 401/14
C07D 403/14
C07D 417/14
C07D 471/04
C07D 473/16
C07D 473/18
C07D 487/04
C07D 495/04
C07D 513/04
A61K 31/4545
A61K 31/52
A61K 31/519
A61P 31/18
European patent
(11) Number of the document 3334723
(13) Kind of document T
(96) European patent application number 16758282.4
Date of filing the European patent application 2016-08-10
(97) Date of publication of the European application 2018-06-20
(45) Date of publication and mention of the grant of the patent 2019-09-18
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/IB2016/054831
Date 2016-08-10
PCT application publication
(87) Number WO 2017/025916
Date 2017-02-16
Priority applications
(30) Number Date Country code
201562203986 P 2015-08-12 US
Inventors
(72)
KADOW, John F., US
NAIDU, B. Narasimhulu, US
WANG, Tao, US
YIN, Zhiwei, US
ZHANG, Zhongxing, US
Grantee
(73) VIIV Healthcare UK (No.5) Limited, 980 Great West Road, Brentford, Middlesex TW8 9GS, GB
Title
(54) 5-(N-[6,5]-FUSED BICYCLIC ARYL TETRAHYDROISOQUINOLIN-6-YL) PYRIDIN-3-YL ACETIC ACID DERIVATIVES AS INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION
  5-(N-[6,5]-FUSED BICYCLIC ARYL TETRAHYDROISOQUINOLIN-6-YL) PYRIDIN-3-YL ACETIC ACID DERIVATIVES AS INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION