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Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
| (51) | INT.CL. | C07D 235/30 | (2006.01) |
| A61P 17/06 | (2018.01) | ||
| C07D 401/04 | (2006.01) | ||
| A61P 3/00 | (2018.01) | ||
| C07D 403/04 | (2006.01) | ||
| C07D 405/04 | (2013.01) | ||
| C07D 405/04 | (2006.01) | ||
| A61P 17/00 | (2018.01) | ||
| C07D 413/04 | (2006.01) | ||
| A61P 13/12 | (2018.01) | ||
| C07D 471/08 | (2006.01) | ||
| A61P 37/02 | (2018.01) | ||
| A61K 31/4184 | (2006.01) | ||
| A61P 19/10 | (2018.01) | ||
| A61P 43/00 | (2018.01) | ||
| A61K 31/4439 | (2006.01) | ||
| A61K 31/506 | (2006.01) | ||
| A61P 9/10 | (2018.01) | ||
| A61P 35/00 | (2006.01) | ||
| C07D 235/30 | (2013.01) | ||
| A61P 25/00 | (2006.01) | ||
| C07D 401/04 | (2013.01) | ||
| A61P 19/00 | (2006.01) | ||
| C07D 471/08 | (2013.01) | ||
| A61P 17/00 | (2006.01) | ||
| C07D 403/04 | (2013.01) | ||
| A61P 3/00 | (2006.01) | ||
| A61K 31/4439 | (2013.01) | ||
| A61P 25/28 | (2018.01) | ||
| A61P 1/00 | (2006.01) | ||
| A61K 31/506 | (2013.01) | ||
| A61P 3/10 | (2018.01) | ||
| A61P 19/00 | (2018.01) | ||
| C07D 451/02 | (2013.01) | ||
| A61P 1/04 | (2018.01) | ||
| C07D 413/04 | (2013.01) | ||
| A61K 31/4184 | (2013.01) | ||
| A61P 29/00 | (2018.01) | ||
| A61P 25/16 | (2018.01) | ||
| A61P 19/06 | (2018.01) | ||
| A61P 25/00 | (2018.01) | ||
| A61P 31/04 | (2018.01) | ||
| A61P 35/00 | (2018.01) | ||
| A61P 19/02 | (2018.01) | ||
| A61P 1/00 | (2018.01) |
| (11) | Patento numeris | 3350170 |
| (13) | Dokumento rūšis | T |
| (96) | Europos patento paraiškos numeris | 16770654.8 |
| Europos patento paraiškos padavimo data | 2016-09-16 | |
| (97) | Europos patento paraiškos paskelbimo data | 2018-07-25 |
| (45) | Paskelbimo apie Europos patento išdavimą data | 2022-01-26 |
| (46) | Apibrėžties vertimo paskelbimo data |
| (86) | Numeris | PCT/US2016/052107 |
| Data | 2016-09-16 |
| (87) | Numeris | WO 2017/049069 |
| Data | 2017-03-23 |
| (30) | Numeris | Data | Šalis |
| 201562220358 P | 2015-09-18 | US |
| (72) |
JORAND-LEBRUN, Catherine , US
LAN, Ruoxi , US
CHEN, Austin , US
CLARK, Ryan C. , US
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| (73) |
Merck Patent GmbH ,
Frankfurter Strasse 250, 64293 Darmstadt,
DE
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| (54) | HETEROARYL COMPOUNDS AS IRAK INHIBITORS AND USES THEREOF |
| HETEROARYL COMPOUNDS AS IRAK INHIBITORS AND USES THEREOF |