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LT - PROCESS FOR THE PREPARATION OF TRICYCLIC PI3K INHIBITOR COMPOUNDS AND METHODS FOR USING THE SAME FOR THE TREATMENT OF CANCER
EN - PROCESS FOR THE PREPARATION OF TRICYCLIC PI3K INHIBITOR COMPOUNDS AND METHODS FOR USING THE SAME FOR THE TREATMENT OF CANCER

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Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. A61K 31/519 (2006.01)
A61K 31/495 (2013.01)
A61K 31/5383 (2006.01)
A61K 31/5383 (2013.01)
C07D 498/14 (2006.01)
A61P 35/00 (2018.01)
C07D 487/04 (2013.01)
C07D 498/14 (2013.01)
C07D 498/22 (2013.01)
European patent
(11) Number of the document 3389662
(13) Kind of document T
(96) European patent application number 16876773.9
Date of filing the European patent application 2016-12-16
(97) Date of publication of the European application 2018-10-24
(45) Date of publication and mention of the grant of the patent 2021-12-01
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2016/067174
Date 2016-12-16
PCT application publication
(87) Number WO 2017/106647
Date 2017-06-22
Priority applications
(30) Number Date Country code
201562268149 P 2015-12-16 US
201662288832 P 2016-01-29 US
201662291248 P 2016-02-04 US
Inventors
(72)
STUMPF, Andreas , US
ANGELAUD, Remy , US
MCCLORY, Andrew , US
YAJIMA, Herbert , US
NDUBAKU, Chudi , US
OLIVERO, Alan , US
Grantee
(73) Genentech, Inc. , 1 DNA Way, South San Francisco, CA 94080, US
Title
(54) PROCESS FOR THE PREPARATION OF TRICYCLIC PI3K INHIBITOR COMPOUNDS AND METHODS FOR USING THE SAME FOR THE TREATMENT OF CANCER
  PROCESS FOR THE PREPARATION OF TRICYCLIC PI3K INHIBITOR COMPOUNDS AND METHODS FOR USING THE SAME FOR THE TREATMENT OF CANCER