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Legal status
Patent not validated
(51) | INT.CL. | A61K 31/519 | (2006.01) |
A61K 31/495 | (2013.01) | ||
A61K 31/5383 | (2006.01) | ||
A61K 31/5383 | (2013.01) | ||
C07D 498/14 | (2006.01) | ||
A61P 35/00 | (2018.01) | ||
C07D 487/04 | (2013.01) | ||
C07D 498/14 | (2013.01) | ||
C07D 498/22 | (2013.01) |
(11) | Number of the document | 3389662 |
(13) | Kind of document | T |
(96) | European patent application number | 16876773.9 |
Date of filing the European patent application | 2016-12-16 | |
(97) | Date of publication of the European application | 2018-10-24 |
(45) | Date of publication and mention of the grant of the patent | 2021-12-01 |
(46) | Date of publication of the claims translation |
(86) | Number | PCT/US2016/067174 |
Date | 2016-12-16 |
(87) | Number | WO 2017/106647 |
Date | 2017-06-22 |
(30) | Number | Date | Country code |
201562268149 P | 2015-12-16 | US | |
201662288832 P | 2016-01-29 | US | |
201662291248 P | 2016-02-04 | US |
(72) |
STUMPF, Andreas , US
ANGELAUD, Remy , US
MCCLORY, Andrew , US
YAJIMA, Herbert , US
NDUBAKU, Chudi , US
OLIVERO, Alan , US
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(73) |
Genentech, Inc. ,
1 DNA Way, South San Francisco, CA 94080,
US
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(54) | PROCESS FOR THE PREPARATION OF TRICYCLIC PI3K INHIBITOR COMPOUNDS AND METHODS FOR USING THE SAME FOR THE TREATMENT OF CANCER |
PROCESS FOR THE PREPARATION OF TRICYCLIC PI3K INHIBITOR COMPOUNDS AND METHODS FOR USING THE SAME FOR THE TREATMENT OF CANCER |