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LT - INTERMEDIATES IN THE SYNTHESIS OF ERIBULIN AND RELATED METHODS OF SYNTHESIS
EN - INTERMEDIATES IN THE SYNTHESIS OF ERIBULIN AND RELATED METHODS OF SYNTHESIS

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Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. A61K 31/35
A61K 31/357
C07D 307/20
C07D 493/04
C07D 493/22
European patent
(11) Number of the document 3413887
(13) Kind of document T
(96) European patent application number 17750887.6
Date of filing the European patent application 2017-02-10
(97) Date of publication of the European application 2018-12-19
(45) Date of publication and mention of the grant of the patent 2021-04-07
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2017/017501
Date 2017-02-10
PCT application publication
(87) Number WO 2017/139664
Date 2017-08-17
Priority applications
(30) Number Date Country code
201662294538 P 2016-02-12 US
Inventors
(72)
BARAN, Phil, S., US
CHASE, Charles, E., US
FANG, Francis, G., US
Grantee
(73) Eisai R&D Management Co., Ltd., 6-10, Koishikawa 4-chome Bunkyo-ku, Tokyo 112-8088, JP
Title
(54) INTERMEDIATES IN THE SYNTHESIS OF ERIBULIN AND RELATED METHODS OF SYNTHESIS
  INTERMEDIATES IN THE SYNTHESIS OF ERIBULIN AND RELATED METHODS OF SYNTHESIS