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LT - EFFICIENT PROCESS FOR THE PREPARATION OF SITAGLIPTIN THROUGH A VERY EFFECTIVE PREPARATION OF THE INTERMEDIATE 2,4,5-TRIFLUOROPHENYLACETIC ACID
EN - EFFICIENT PROCESS FOR THE PREPARATION OF SITAGLIPTIN THROUGH A VERY EFFECTIVE PREPARATION OF THE INTERMEDIATE 2,4,5-TRIFLUOROPHENYLACETIC ACID

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 487/04
European patent
(11) Number of the document 3424927
(13) Kind of document T
(96) European patent application number 17179524.8
Date of filing the European patent application 2017-07-04
(97) Date of publication of the European application 2019-01-09
(45) Date of publication and mention of the grant of the patent 2019-04-17
(46) Date of publication of the claims translation
Inventors
(72)
De Lucchi, Ottorino, IT
Padovan, Pierluigi, IT
Brasola, Elena, IT
Grantee
(73) F.I.S.- Fabbrica Italiana Sintetici S.p.A., Viale Milano, 26, 36075 Montecchio Maggiore (VI), IT
Title
(54) EFFICIENT PROCESS FOR THE PREPARATION OF SITAGLIPTIN THROUGH A VERY EFFECTIVE PREPARATION OF THE INTERMEDIATE 2,4,5-TRIFLUOROPHENYLACETIC ACID
  EFFICIENT PROCESS FOR THE PREPARATION OF SITAGLIPTIN THROUGH A VERY EFFECTIVE PREPARATION OF THE INTERMEDIATE 2,4,5-TRIFLUOROPHENYLACETIC ACID