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LT - AROMATIC RING COMPOUND HAVING A CHOLINERGIC MUSCARINE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATOR ACTIVITY
EN - AROMATIC RING COMPOUND HAVING A CHOLINERGIC MUSCARINE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATOR ACTIVITY

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 405/14 (2013.01)
C07D 213/56 (2006.01)
A61K 31/415 (2006.01)
A61K 31/415 (2013.01)
A61K 31/427 (2013.01)
A61K 31/4192 (2006.01)
A61K 31/4406 (2013.01)
A61K 31/427 (2006.01)
A61K 31/4406 (2006.01)
A61K 31/4439 (2013.01)
A61K 31/4439 (2006.01)
C07D 231/12 (2013.01)
A61P 25/04 (2006.01)
C07D 401/04 (2013.01)
A61P 25/16 (2006.01)
C07D 405/12 (2013.01)
A61P 25/18 (2006.01)
C07D 413/12 (2013.01)
C07D 417/12 (2013.01)
A61P 25/20 (2006.01)
C07D 249/06 (2013.01)
A61P 25/28 (2006.01)
C07D 213/56 (2013.01)
C07D 231/12 (2006.01)
C07D 249/06 (2006.01)
A61K 31/4192 (2013.01)
C07D 401/04 (2006.01)
A61P 25/20 (2018.01)
C07D 405/12 (2006.01)
A61P 25/28 (2018.01)
C07D 405/14 (2006.01)
A61P 25/18 (2018.01)
A61P 25/16 (2018.01)
C07D 413/12 (2006.01)
A61K 31/4155 (2013.01)
C07D 417/12 (2006.01)
A61K 31/4155 (2006.01)
European patent
(11) Number of the document 3428150
(13) Kind of document T
(96) European patent application number 17763390.6
Date of filing the European patent application 2017-03-09
(97) Date of publication of the European application 2019-01-16
(45) Date of publication and mention of the grant of the patent 2023-07-12
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/JP2017/009529
Date 2017-03-09
PCT application publication
(87) Number WO 2017/155050
Date 2017-09-14
Priority applications
(30) Number Date Country code
2016048866 2016-03-11 JP
2016134234 2016-07-06 JP
Inventors
(72)
OGINO, Masaki , JP
KIMURA, Eiji , JP
SUZUKI, Shinkichi , JP
FUJI, Kouji , JP
OHASHI, Tomohiro , JP
FUSHIMI, Makoto , JP
MASUDA, Kei , JP
KOIKE, Tatsuki , JP
WAKABAYASHI, Takeshi , JP
YONEMORI, Jinichi , JP
YAMADA, Masami , JP
Grantee
(73) Takeda Pharmaceutical Company Limited , 1-1 Doshomachi 4-chome Chuo-ku, Osaka-shi, Osaka 541-0045, JP
Title
(54) AROMATIC RING COMPOUND HAVING A CHOLINERGIC MUSCARINE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATOR ACTIVITY
  AROMATIC RING COMPOUND HAVING A CHOLINERGIC MUSCARINE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATOR ACTIVITY