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LT - PROCESS AND INTERMEDIATES FOR PREPARING PRODRUGS OF PYRIDONE AMIDES USEFUL AS MODULATORS OF SODIUM CHANNELS
EN - PROCESS AND INTERMEDIATES FOR PREPARING PRODRUGS OF PYRIDONE AMIDES USEFUL AS MODULATORS OF SODIUM CHANNELS

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07F 9/576 (2013.01)
C07F 9/576 (2006.01)
C07F 9/58 (2006.01)
C07F 9/58 (2013.01)
A61P 1/00 (2018.01)
A61P 1/02 (2018.01)
A61P 1/06 (2018.01)
A61P 11/14 (2018.01)
A61P 13/00 (2018.01)
A61P 13/02 (2018.01)
A61P 19/00 (2018.01)
A61P 19/02 (2018.01)
A61P 21/00 (2018.01)
A61P 25/00 (2018.01)
A61P 25/02 (2018.01)
A61P 25/04 (2018.01)
A61P 29/00 (2018.01)
A61P 43/00 (2018.01)
A61P 9/06 (2018.01)
European patent
(11) Number of the document 3459958
(13) Kind of document T
(96) European patent application number 18186616.1
Date of filing the European patent application 2014-12-12
(97) Date of publication of the European application 2019-03-27
(45) Date of publication and mention of the grant of the patent 2024-08-07
(46) Date of publication of the claims translation
Priority applications
(30) Number Date Country code
201361915937 P 2013-12-13 US
Inventors
(72)
ANDERSON, Corey , US
HADIDA-RUAH, Sara Sabina , US
GOLEC, Julian Marian Charles , GB
ZHANG, Beili , US
LITTLER, Benjamin Joseph , US
KESHAVARZ-SHOKRI, Ali , US
ALCACIO, Tim Edward , US
BELMONT, Daniel T. , US
Grantee
(73) Vertex Pharmaceuticals Incorporated , 50 Northern Avenue, Boston, MA 02210, US
Title
(54) PROCESS AND INTERMEDIATES FOR PREPARING PRODRUGS OF PYRIDONE AMIDES USEFUL AS MODULATORS OF SODIUM CHANNELS
  PROCESS AND INTERMEDIATES FOR PREPARING PRODRUGS OF PYRIDONE AMIDES USEFUL AS MODULATORS OF SODIUM CHANNELS