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EN | LT
LT - (S)-4-(8-AMINO-3-(1-(BUT-2-YNOYL)PYRROLIDIN-2-YL)IMIDAZO[1,5-A]PYRAZIN-1-YL)-2-METHOXY-N-(PYRIDIN-2-YL)BENZAMIDE AS BTK-INHIBITOR
EN - (S)-4-(8-AMINO-3-(1-(BUT-2-YNOYL)PYRROLIDIN-2-YL)IMIDAZO[1,5-A]PYRAZIN-1-YL)-2-METHOXY-N-(PYRIDIN-2-YL)BENZAMIDE AS BTK-INHIBITOR

Teisinis statusas

Patentas neįsigaliojo (pagal EPK)

Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) INT.CL. C07D 487/04 (2006.01)
C07D 519/00 (2013.01)
C07D 519/00 (2006.01)
C07D 487/04 (2013.01)
A61K 31/4985 (2006.01)
A61P 1/00 (2018.01)
A61P 19/08 (2006.01)
A61P 1/02 (2018.01)
A61P 29/00 (2006.01)
A61P 1/04 (2018.01)
A61P 31/00 (2006.01)
A61P 1/16 (2018.01)
A61P 35/00 (2006.01)
A61P 1/18 (2018.01)
A61P 37/00 (2006.01)
A61P 11/00 (2018.01)
A61P 11/06 (2018.01)
A61P 13/02 (2018.01)
A61P 13/12 (2018.01)
A61P 17/00 (2018.01)
A61P 17/06 (2018.01)
A61P 19/00 (2018.01)
A61P 19/02 (2018.01)
A61P 19/08 (2018.01)
A61P 21/04 (2018.01)
A61P 25/00 (2018.01)
A61P 27/02 (2018.01)
A61P 27/06 (2018.01)
A61P 27/16 (2018.01)
A61P 29/00 (2018.01)
A61P 31/00 (2018.01)
A61P 31/04 (2018.01)
A61P 31/12 (2018.01)
A61P 35/00 (2018.01)
A61P 35/02 (2018.01)
A61P 37/00 (2018.01)
A61P 37/02 (2018.01)
A61P 37/06 (2018.01)
A61P 43/00 (2018.01)
A61P 5/14 (2018.01)
A61P 7/00 (2018.01)
A61P 7/06 (2018.01)
A61P 3/10 (2018.01)
Europos patentas
(11) Patento numeris 3495368
(13) Dokumento rūšis T
(96) Europos patento paraiškos numeris 18203086.6
Europos patento paraiškos padavimo data 2012-07-11
(97) Europos patento paraiškos paskelbimo data 2019-06-12
(45) Paskelbimo apie Europos patento išdavimą data 2023-05-31
(46) Apibrėžties vertimo paskelbimo data
Prioriteto paraiškos
(30) Numeris Data Šalis
201161509397 P 2011-07-19 US
11174578 2011-07-19 EP
Išradėjai
(72)
BARF, Tjeerd A. , NL
JANS, Christiaan Geradus Johannes Maria , NL
de MAN, Adrianus Petrus Antonius , NL
OUBRIE, Arthur A. , NL
RAAIJMAKERS, Hans C.A. , NL
REWINKEL, Johannes Bernardus Maria , NL
STERRENBURG, Jan-Gerard , NL
WIJKMANS, Jacobus C.H.M. , NL
Savininkas
(73) Merck Sharp & Dohme B.V. , Waarderweg 39, 2031 BN Haarlem, NL
Pavadinimas
(54) (S)-4-(8-AMINO-3-(1-(BUT-2-YNOYL)PYRROLIDIN-2-YL)IMIDAZO[1,5-A]PYRAZIN-1-YL)-2-METHOXY-N-(PYRIDIN-2-YL)BENZAMIDE AS BTK-INHIBITOR
  (S)-4-(8-AMINO-3-(1-(BUT-2-YNOYL)PYRROLIDIN-2-YL)IMIDAZO[1,5-A]PYRAZIN-1-YL)-2-METHOXY-N-(PYRIDIN-2-YL)BENZAMIDE AS BTK-INHIBITOR