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Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
| (51) | INT.CL. | C07D 487/04 | (2006.01) |
| C07D 519/00 | (2013.01) | ||
| C07D 519/00 | (2006.01) | ||
| C07D 487/04 | (2013.01) | ||
| A61K 31/4985 | (2006.01) | ||
| A61P 1/00 | (2018.01) | ||
| A61P 19/08 | (2006.01) | ||
| A61P 1/02 | (2018.01) | ||
| A61P 29/00 | (2006.01) | ||
| A61P 1/04 | (2018.01) | ||
| A61P 31/00 | (2006.01) | ||
| A61P 1/16 | (2018.01) | ||
| A61P 35/00 | (2006.01) | ||
| A61P 1/18 | (2018.01) | ||
| A61P 37/00 | (2006.01) | ||
| A61P 11/00 | (2018.01) | ||
| A61P 11/06 | (2018.01) | ||
| A61P 13/02 | (2018.01) | ||
| A61P 13/12 | (2018.01) | ||
| A61P 17/00 | (2018.01) | ||
| A61P 17/06 | (2018.01) | ||
| A61P 19/00 | (2018.01) | ||
| A61P 19/02 | (2018.01) | ||
| A61P 19/08 | (2018.01) | ||
| A61P 21/04 | (2018.01) | ||
| A61P 25/00 | (2018.01) | ||
| A61P 27/02 | (2018.01) | ||
| A61P 27/06 | (2018.01) | ||
| A61P 27/16 | (2018.01) | ||
| A61P 29/00 | (2018.01) | ||
| A61P 31/00 | (2018.01) | ||
| A61P 31/04 | (2018.01) | ||
| A61P 31/12 | (2018.01) | ||
| A61P 35/00 | (2018.01) | ||
| A61P 35/02 | (2018.01) | ||
| A61P 37/00 | (2018.01) | ||
| A61P 37/02 | (2018.01) | ||
| A61P 37/06 | (2018.01) | ||
| A61P 43/00 | (2018.01) | ||
| A61P 5/14 | (2018.01) | ||
| A61P 7/00 | (2018.01) | ||
| A61P 7/06 | (2018.01) | ||
| A61P 3/10 | (2018.01) |
| (11) | Patento numeris | 3495368 |
| (13) | Dokumento rūšis | T |
| (96) | Europos patento paraiškos numeris | 18203086.6 |
| Europos patento paraiškos padavimo data | 2012-07-11 | |
| (97) | Europos patento paraiškos paskelbimo data | 2019-06-12 |
| (45) | Paskelbimo apie Europos patento išdavimą data | 2023-05-31 |
| (46) | Apibrėžties vertimo paskelbimo data |
| (30) | Numeris | Data | Šalis |
| 201161509397 P | 2011-07-19 | US | |
| 11174578 | 2011-07-19 | EP |
| (72) |
BARF, Tjeerd A. , NL
JANS, Christiaan Geradus Johannes Maria , NL
de MAN, Adrianus Petrus Antonius , NL
OUBRIE, Arthur A. , NL
RAAIJMAKERS, Hans C.A. , NL
REWINKEL, Johannes Bernardus Maria , NL
STERRENBURG, Jan-Gerard , NL
WIJKMANS, Jacobus C.H.M. , NL
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| (73) |
Merck Sharp & Dohme B.V. ,
Waarderweg 39, 2031 BN Haarlem,
NL
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| (54) | (S)-4-(8-AMINO-3-(1-(BUT-2-YNOYL)PYRROLIDIN-2-YL)IMIDAZO[1,5-A]PYRAZIN-1-YL)-2-METHOXY-N-(PYRIDIN-2-YL)BENZAMIDE AS BTK-INHIBITOR |
| (S)-4-(8-AMINO-3-(1-(BUT-2-YNOYL)PYRROLIDIN-2-YL)IMIDAZO[1,5-A]PYRAZIN-1-YL)-2-METHOXY-N-(PYRIDIN-2-YL)BENZAMIDE AS BTK-INHIBITOR |