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LT - PROCESS AND INTERMEDIATES FOR THE PREPARATION OF NAPHTHYRIDINE COMPOUNDS AS JAK KINASE INHIBITORS
EN - PROCESS AND INTERMEDIATES FOR THE PREPARATION OF NAPHTHYRIDINE COMPOUNDS AS JAK KINASE INHIBITORS

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 519/00 (2006.01)
C07D 519/00 (2013.01)
A61K 31/439 (2006.01)
A61K 31/46 (2013.01)
A61P 1/04 (2006.01)
A61P 1/00 (2018.01)
A61P 1/04 (2018.01)
A61P 29/00 (2018.01)
A61P 43/00 (2018.01)
European patent
(11) Number of the document 3569604
(13) Kind of document T
(96) European patent application number 19182836.7
Date of filing the European patent application 2016-05-26
(97) Date of publication of the European application 2019-11-20
(45) Date of publication and mention of the grant of the patent 2022-07-06
(46) Date of publication of the claims translation
Priority applications
(30) Number Date Country code
201562167694 P 2015-05-28 US
201662312273 P 2016-03-23 US
Inventors
(72)
HUDSON, Ryan , US
KOZAK, Jennifer , US
FATHEREE, Paul R , US
PODESTO, Dante D , US
BRANDT, Gary E.L. , US
FLEURY, Melissa , US
BEAUSOLEIL, Anne-Marie , US
HUANG, Xiaojun , US
THALLADI, Venkat R. , US
Grantee
(73) Theravance Biopharma R&D IP, LLC , 901 Gateway Boulevard, South San Francisco, CA 94080, US
Title
(54) PROCESS AND INTERMEDIATES FOR THE PREPARATION OF NAPHTHYRIDINE COMPOUNDS AS JAK KINASE INHIBITORS
  PROCESS AND INTERMEDIATES FOR THE PREPARATION OF NAPHTHYRIDINE COMPOUNDS AS JAK KINASE INHIBITORS