LT - A CRYSTALLINE FORM OF (S) 2 ETHYLBUTYL 2 (((S) (((2R,3S,4R,5R) 5 (4 AMINOPYRROLO[2,1-F][1,2,4]TRIAZIN-7-YL)-5-CYANO-3,4-DIHYDROXYTETRAHYDROFURAN-2 YL)METHOXY)(PHENOXY) PHOSPHORYL)AMINO)PROPANOATE
EN - A CRYSTALLINE FORM OF (S) 2 ETHYLBUTYL 2 (((S) (((2R,3S,4R,5R) 5 (4 AMINOPYRROLO[2,1-F][1,2,4]TRIAZIN-7-YL)-5-CYANO-3,4-DIHYDROXYTETRAHYDROFURAN-2 YL)METHOXY)(PHENOXY) PHOSPHORYL)AMINO)PROPANOATE
Legal status
Patent not validated
Bibliographic data
Indications of the International Patent Classification (IPC)
| (51) |
INT.CL. |
C07F 9/6561 |
(2006.01) |
|
|
C07F 9/6561 |
(2013.01) |
|
|
A61P 31/14 |
(2006.01) |
|
|
A61P 31/14 |
(2018.01) |
|
|
A61K 31/53 |
(2006.01) |
|
|
C07H 19/00 |
(2013.01) |
|
|
Y02A 50/30 |
(2018.01) |
European patent
| (11) |
Number of the document |
3618929 |
| (13) |
Kind of document |
T |
| (96) |
European patent application number |
18724731.7 |
|
Date of filing the European patent application |
2018-04-27 |
| (97) |
Date of publication of the European application |
2020-03-11 |
| (45) |
Date of publication and mention of the grant of the patent |
2022-12-07
|
| (46) |
Date of publication of the claims translation |
|
PCT application
| (86) |
Number |
PCT/US2018/029974 |
|
Date |
2018-04-27 |
PCT application publication
| (87) |
Number |
WO 2018/204198 |
|
Date |
2018-11-08 |
Priority applications
| (30) |
Number |
Date |
Country code |
|
201762492364 P |
2017-05-01
|
US |
Inventors
| (72) |
BRAK, Katrien , US
CARRA, Ernest A. , US
HEUMANN, Lars V. , US
LARSON, Nate , US
|
Grantee
| (73) |
Gilead Sciences, Inc. ,
333 Lakeside Drive, Foster City, CA 94404,
US
|
Title
| (54) |
A CRYSTALLINE FORM OF (S) 2 ETHYLBUTYL 2 (((S) (((2R,3S,4R,5R) 5 (4 AMINOPYRROLO[2,1-F][1,2,4]TRIAZIN-7-YL)-5-CYANO-3,4-DIHYDROXYTETRAHYDROFURAN-2 YL)METHOXY)(PHENOXY) PHOSPHORYL)AMINO)PROPANOATE |
| |
A CRYSTALLINE FORM OF (S) 2 ETHYLBUTYL 2 (((S) (((2R,3S,4R,5R) 5 (4 AMINOPYRROLO[2,1-F][1,2,4]TRIAZIN-7-YL)-5-CYANO-3,4-DIHYDROXYTETRAHYDROFURAN-2 YL)METHOXY)(PHENOXY) PHOSPHORYL)AMINO)PROPANOATE |