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LT - PROCESS FOR PREPARING AN INTERMEDIATE IN THE SYNTHESIS OF (CYCLOPENTYL[D]PYRIMIDIN-4-YL)PIPERAZINE COMPOUNDS
EN - PROCESS FOR PREPARING AN INTERMEDIATE IN THE SYNTHESIS OF (CYCLOPENTYL[D]PYRIMIDIN-4-YL)PIPERAZINE COMPOUNDS

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Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 239/46 (2006.01)
C12Y 305/05001 (2013.01)
Y02P 20/55 (2015.11)
C07D 239/42 (2013.01)
C07D 239/70 (2013.01)
C12N 9/78 (2013.01)
C07D 239/46 (2013.01)
C07D 239/54 (2013.01)
European patent
(11) Number of the document 3626710
(13) Kind of document T
(96) European patent application number 19191353.2
Date of filing the European patent application 2015-09-25
(97) Date of publication of the European application 2020-03-25
(45) Date of publication and mention of the grant of the patent 2022-02-16
(46) Date of publication of the claims translation
Priority applications
(30) Number Date Country code
201462055893 P 2014-09-26 US
Inventors
(72)
GOSSELIN, Francis , US
HAN, Chong , US
IDING, Hans , CH
REENTS, Reinhard , CH
SAVAGE, Scott , US
WIRZ, Beat , CH
Grantee
(73) F. Hoffmann-La Roche AG , Grenzacherstrasse 124, 4070 Basel, CH
GENENTECH, INC. , 1 DNA Way, South San Francisco, CA 94080-4990, US
Title
(54) PROCESS FOR PREPARING AN INTERMEDIATE IN THE SYNTHESIS OF (CYCLOPENTYL[D]PYRIMIDIN-4-YL)PIPERAZINE COMPOUNDS
  PROCESS FOR PREPARING AN INTERMEDIATE IN THE SYNTHESIS OF (CYCLOPENTYL[D]PYRIMIDIN-4-YL)PIPERAZINE COMPOUNDS