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LT - CRYSTALLINE SOLID FORMS OF SALTS OF N-{4-[(6,7-DIMETHOXYQUINOLIN-4-YL) OXY]PHENYL}-N'-(4-FLUORPHENYL) CYCLOPROPANE-1,1-DICARBOXAMIDE, PROCESSES FOR MAKING, AND METHODS OF USE
EN - CRYSTALLINE SOLID FORMS OF SALTS OF N-{4-[(6,7-DIMETHOXYQUINOLIN-4-YL) OXY]PHENYL}-N'-(4-FLUORPHENYL) CYCLOPROPANE-1,1-DICARBOXAMIDE, PROCESSES FOR MAKING, AND METHODS OF USE

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 215/22 (2006.01)
C07D 215/22 (2013.01)
A61K 31/47 (2006.01)
A61P 35/00 (2018.01)
A61P 35/00 (2006.01)
European patent
(11) Number of the document 3630726
(13) Kind of document T
(96) European patent application number 18732548.5
Date of filing the European patent application 2018-05-26
(97) Date of publication of the European application 2020-04-08
(45) Date of publication and mention of the grant of the patent 2021-12-22
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2018/034784
Date 2018-05-26
PCT application publication
(87) Number WO 2018/218233
Date 2018-11-29
Priority applications
(30) Number Date Country code
201762511714 P 2017-05-26 US
Inventors
(72)
SHAH, Khalid , US
Grantee
(73) Exelixis, Inc. , 1851 Harbor Bay Parkway, Alameda, CA 94502, US
Title
(54) CRYSTALLINE SOLID FORMS OF SALTS OF N-{4-[(6,7-DIMETHOXYQUINOLIN-4-YL) OXY]PHENYL}-N'-(4-FLUORPHENYL) CYCLOPROPANE-1,1-DICARBOXAMIDE, PROCESSES FOR MAKING, AND METHODS OF USE
  CRYSTALLINE SOLID FORMS OF SALTS OF N-{4-[(6,7-DIMETHOXYQUINOLIN-4-YL) OXY]PHENYL}-N'-(4-FLUORPHENYL) CYCLOPROPANE-1,1-DICARBOXAMIDE, PROCESSES FOR MAKING, AND METHODS OF USE