LT - MODIFIED NUCLEIC ACID MONOMERS AND OLIGONUCLEIC ACID ANALOGUES, WITH HIGH BIOLOGICAL STABILITY AND TARGET GENE SILENCING ACTIVITY, FOR USE IN THERAPY AND DIAGNOSIS OF CANCER AND VIRAL DISEASES
EN - MODIFIED NUCLEIC ACID MONOMERS AND OLIGONUCLEIC ACID ANALOGUES, WITH HIGH BIOLOGICAL STABILITY AND TARGET GENE SILENCING ACTIVITY, FOR USE IN THERAPY AND DIAGNOSIS OF CANCER AND VIRAL DISEASES
Legal status
Patent not validated
Bibliographic data
Indications of the International Patent Classification (IPC)
(51) |
INT.CL. |
A61P 31/12 |
(2018.01) |
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C07D 239/54 |
(2006.01) |
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C07F 7/18 |
(2006.01) |
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A61P 35/00 |
(2018.01) |
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C07D 239/54 |
(2013.01) |
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C07F 9/6512 |
(2006.01) |
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C07F 9/6512 |
(2013.01) |
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C07F 9/6561 |
(2006.01) |
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C07H 21/02 |
(2013.01) |
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C07H 21/02 |
(2006.01) |
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A61K 9/00 |
(2006.01) |
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C07F 9/65616 |
(2013.01) |
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A61K 9/1271 |
(2013.01) |
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A61K 9/08 |
(2006.01) |
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A61K 9/0019 |
(2013.01) |
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A61K 9/127 |
(2006.01) |
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C12N 15/88 |
(2013.01) |
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A61K 31/513 |
(2006.01) |
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C12N2310/14 |
(2013.01) |
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A61K 31/713 |
(2006.01) |
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C12N 15/113 |
(2013.01) |
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A61K 48/00 |
(2006.01) |
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C12N2310/323 |
(2013.01) |
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A61P 31/12 |
(2006.01) |
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C12N2310/322 |
(2013.01) |
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A61P 35/00 |
(2006.01) |
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Y02P 20/55 |
(2015.11) |
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C12N 15/00 |
(2006.01) |
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C12N 15/88 |
(2006.01) |
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C12N 15/113 |
(2010.01) |
European patent
(11) |
Number of the document |
3643706 |
(13) |
Kind of document |
T |
(96) |
European patent application number |
18817223.3 |
|
Date of filing the European patent application |
2018-06-14 |
(97) |
Date of publication of the European application |
2020-04-29 |
(45) |
Date of publication and mention of the grant of the patent |
2023-11-15
|
(46) |
Date of publication of the claims translation |
|
PCT application
(86) |
Number |
PCT/JP2018/022663 |
|
Date |
2018-06-14 |
PCT application publication
(87) |
Number |
WO 2018/230624 |
|
Date |
2018-12-20 |
Priority applications
(30) |
Number |
Date |
Country code |
|
2017118572 |
2017-06-16
|
JP |
Inventors
(72) |
TAKAHASHI Yoshinori , JP
SUZUKI Yuta , JP
|
Grantee
(73) |
Eisai R&D Management Co., Ltd. ,
4-6-10 Koishikawa
Bunkyo-ku, Tokyo 112-8088,
JP
|
Title
(54) |
MODIFIED NUCLEIC ACID MONOMERS AND OLIGONUCLEIC ACID ANALOGUES, WITH HIGH BIOLOGICAL STABILITY AND TARGET GENE SILENCING ACTIVITY, FOR USE IN THERAPY AND DIAGNOSIS OF CANCER AND VIRAL DISEASES |
|
MODIFIED NUCLEIC ACID MONOMERS AND OLIGONUCLEIC ACID ANALOGUES, WITH HIGH BIOLOGICAL STABILITY AND TARGET GENE SILENCING ACTIVITY, FOR USE IN THERAPY AND DIAGNOSIS OF CANCER AND VIRAL DISEASES |