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LT - N-((1R,2S,SR)-5-(tret-butilamino)-2-((S)-3-(7-tret-butilpirazolo[1,5-a][1,3,5]triazin-4-ilamino)-2-oksopirolidin-1-il)cikloheksil)acetamido gamybos būdas
EN - PROCESS FOR THE PREPARATION OF N-((1R,2S,SR)-5-(TERT-BUTYLAMINO)-2-((S)-3-(7-TERT-BUTYLPYRAZOLO[1,5-A][1,3,5]TRIAZIN-4-YLAMINO)-2-OXOPYRROLIDIN-1-YL)CYCLOHEXYL)ACETAMIDE

Legal status

Patent lapsed (non-payment of fees)

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 235/06 (2006.01)
C07C 233/41 (2006.01)
C07D 487/04 (2006.01)
C07D 207/273 (2006.01)
European patent
(11) Number of the document 3655395
(13) Kind of document T
(96) European patent application number 18785785.9
Date of filing the European patent application 2018-07-19
(97) Date of publication of the European application 2020-05-27
(45) Date of publication and mention of the grant of the patent 2021-12-01
(46) Date of publication of the claims translation 2022-03-10
PCT application
(86) Number PCT/US2018/042797
Date 2018-07-19
PCT application publication
(87) Number WO 2019/018592
Date 2019-01-24
Priority applications
(30) Number Date Country code
201762534908 P 2017-07-20 US
Inventors
(72)
AYTAR, Burcu Selin , US
BOROVIKA, Alina , US
CHAN, Collin , US
DEERBERG, Joerg , US
DOMAGALSKI, Nathan R. , US
EASTGATE, Martin D. , US
FAN, Yu , US
FENSTER, Michael David Bengt , US
FOREST, Robert V. , US
GONZALEZ-BOBES, Francisco , US
GREEN, Rebecca A. , US
HICKEY, Matthew R. , US
KOPP, Nathaniel David , US
LA CRUZ, Thomas E. , US
LAUSER, Kathleen , US
LEE, Hong Geun , KR
LEAHY, David K. , US
LUO, Helen Y. , US
RAZLER, Thomas M. , US
SAVAGE, Scott A. , US
SFOUGGATAKIS, Chris , US
SOUMEILLANT, Maxime C.D. , US
ZARETSKY, Serge , US
ZHENG, Bin , US
ZHU, Ye , SG
Grantee
(73) Bristol-Myers Squibb Company , Route 206 and Province Line Road, Princeton, NJ 08543, US
Attorney or representative
(74) Jurga PETNIŪNAITĖ, AAA Law, A. Goštauto g. 40B, Verslo centras "Dvyniai", LT-03163 Vilnius, LT
Title
(54) N-((1R,2S,SR)-5-(tret-butilamino)-2-((S)-3-(7-tret-butilpirazolo[1,5-a][1,3,5]triazin-4-ilamino)-2-oksopirolidin-1-il)cikloheksil)acetamido gamybos būdas
  PROCESS FOR THE PREPARATION OF N-((1R,2S,SR)-5-(TERT-BUTYLAMINO)-2-((S)-3-(7-TERT-BUTYLPYRAZOLO[1,5-A][1,3,5]TRIAZIN-4-YLAMINO)-2-OXOPYRROLIDIN-1-YL)CYCLOHEXYL)ACETAMIDE
Last renewal fee
Payment date Validity (years) Amount
2023-07-03 6 139.00 EUR
Legal status
Patent lapsed (non-payment of fees)
Invalidation date 2024-07-19