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LT - N-HETEROCYCLIC COMPOUNDS AS OREXIN 2 AGONISTS FOR THE TREATMENT OF NEUROLOGICAL DISORDERS
EN - N-HETEROCYCLIC COMPOUNDS AS OREXIN 2 AGONISTS FOR THE TREATMENT OF NEUROLOGICAL DISORDERS

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 405/06 (2013.01)
C07D 211/36 (2006.01)
C07D 401/06 (2006.01)
C07D 211/36 (2013.01)
A61P 25/00 (2018.01)
C07D 405/06 (2006.01)
C07D 205/04 (2013.01)
C07D 417/06 (2006.01)
C07D 205/04 (2006.01)
C07D 207/14 (2013.01)
C07D 207/14 (2006.01)
C07D 211/56 (2013.01)
C07D 211/56 (2006.01)
C07D 401/06 (2013.01)
C07D 401/10 (2006.01)
C07D 401/10 (2013.01)
C07D 401/14 (2006.01)
C07D 401/14 (2013.01)
C07D 403/06 (2006.01)
C07D 403/06 (2013.01)
C07D 405/10 (2006.01)
C07D 405/10 (2013.01)
C07D 405/12 (2006.01)
C07D 405/12 (2013.01)
C07D 413/06 (2013.01)
C07D 413/06 (2006.01)
C07D 417/06 (2013.01)
C07D 417/14 (2006.01)
C07D 417/14 (2013.01)
A61P 25/00 (2006.01)
A61K 31/435 (2006.01)
European patent
(11) Number of the document 3661923
(13) Kind of document T
(96) European patent application number 18762939.9
Date of filing the European patent application 2018-08-02
(97) Date of publication of the European application 2020-06-10
(45) Date of publication and mention of the grant of the patent 2024-05-15
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/JP2018/029696
Date 2018-08-02
PCT application publication
(87) Number WO 2019/027058
Date 2019-02-07
Priority applications
(30) Number Date Country code
2017150685 2017-08-03 JP
2017248495 2017-12-25 JP
Inventors
(72)
KAJITA, Yuichi , JP
MIKAMI, Satoshi , JP
MIYANOHANA, Yuhei , JP
KOIKE, Tatsuki , JP
DAINI, Masaki , JP
OYABU, Norio , JP
OGINO, Masaki , JP
TAKEUCHI, Kohei , JP
ITO, Yoshiteru , JP
TOKUNAGA, Norihito , JP
SUGIMOTO, Takahiro , JP
MIYAZAKI,Tohru , JP
ODA, Tsuneo , JP
HOASHI, Yasutaka , JP
HATTORI,Yasushi , JP
IMAMURA, Keisuke , JP
Grantee
(73) Takeda Pharmaceutical Company Limited , 1-1 Doshomachi 4-chome Chuo-ku, Osaka-shi, Osaka 541-0045, JP
Title
(54) N-HETEROCYCLIC COMPOUNDS AS OREXIN 2 AGONISTS FOR THE TREATMENT OF NEUROLOGICAL DISORDERS
  N-HETEROCYCLIC COMPOUNDS AS OREXIN 2 AGONISTS FOR THE TREATMENT OF NEUROLOGICAL DISORDERS