LT - CRYSTALLINE FORMS OF ETHYL ((S)-((((2R,5R)-5-(6-AMINO-9H-PURIN-9-YL)-4-FLUORO-2,5-DIHYDROFURAN-2-YL)OXY)METHYL)(PHENOXY)PHOSPHORYL)-L-ALANINATE (GS-9131) FOR TREATING VIRAL INFECTIONS
EN - CRYSTALLINE FORMS OF ETHYL ((S)-((((2R,5R)-5-(6-AMINO-9H-PURIN-9-YL)-4-FLUORO-2,5-DIHYDROFURAN-2-YL)OXY)METHYL)(PHENOXY)PHOSPHORYL)-L-ALANINATE (GS-9131) FOR TREATING VIRAL INFECTIONS
Legal status
Patent not validated
Bibliographic data
Indications of the International Patent Classification (IPC)
(51) |
INT.CL. |
C07D 473/34 |
(2006.01) |
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C07D 417/12 |
(2006.01) |
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C07D 493/04 |
(2006.01) |
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C07D 498/14 |
(2006.01) |
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A61K 31/5365 |
(2006.01) |
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A61K 31/635 |
(2006.01) |
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A61K 31/5377 |
(2006.01) |
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A61K 31/675 |
(2006.01) |
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A61P 31/18 |
(2006.01) |
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C07H 19/16 |
(2006.01) |
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C07H 19/20 |
(2006.01) |
European patent
(11) |
Number of the document |
3661937 |
(13) |
Kind of document |
T |
(96) |
European patent application number |
18755368.0 |
|
Date of filing the European patent application |
2018-07-30 |
(97) |
Date of publication of the European application |
2020-06-10 |
(45) |
Date of publication and mention of the grant of the patent |
2021-07-28
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(46) |
Date of publication of the claims translation |
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PCT application
(86) |
Number |
PCT/US2018/044415 |
|
Date |
2018-07-30 |
PCT application publication
(87) |
Number |
WO 2019/027920 |
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Date |
2019-02-07 |
Priority applications
(30) |
Number |
Date |
Country code |
|
201762539822 P |
2017-08-01
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US |
Inventors
(72) |
LAPINA, Olga Viktorovna , US
SHI, Bing , US
WANG, Silas , US
|
Grantee
(73) |
Gilead Sciences, Inc. ,
333 Lakeside Drive, Foster City, CA 94404,
US
|
Title
(54) |
CRYSTALLINE FORMS OF ETHYL ((S)-((((2R,5R)-5-(6-AMINO-9H-PURIN-9-YL)-4-FLUORO-2,5-DIHYDROFURAN-2-YL)OXY)METHYL)(PHENOXY)PHOSPHORYL)-L-ALANINATE (GS-9131) FOR TREATING VIRAL INFECTIONS |
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CRYSTALLINE FORMS OF ETHYL ((S)-((((2R,5R)-5-(6-AMINO-9H-PURIN-9-YL)-4-FLUORO-2,5-DIHYDROFURAN-2-YL)OXY)METHYL)(PHENOXY)PHOSPHORYL)-L-ALANINATE (GS-9131) FOR TREATING VIRAL INFECTIONS |