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LT - CRYSTALLINE FORMS OF ETHYL ((S)-((((2R,5R)-5-(6-AMINO-9H-PURIN-9-YL)-4-FLUORO-2,5-DIHYDROFURAN-2-YL)OXY)METHYL)(PHENOXY)PHOSPHORYL)-L-ALANINATE (GS-9131) FOR TREATING VIRAL INFECTIONS
EN - CRYSTALLINE FORMS OF ETHYL ((S)-((((2R,5R)-5-(6-AMINO-9H-PURIN-9-YL)-4-FLUORO-2,5-DIHYDROFURAN-2-YL)OXY)METHYL)(PHENOXY)PHOSPHORYL)-L-ALANINATE (GS-9131) FOR TREATING VIRAL INFECTIONS

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 473/34 (2006.01)
C07D 417/12 (2006.01)
C07D 493/04 (2006.01)
C07D 498/14 (2006.01)
A61K 31/5365 (2006.01)
A61K 31/635 (2006.01)
A61K 31/5377 (2006.01)
A61K 31/675 (2006.01)
A61P 31/18 (2006.01)
C07H 19/16 (2006.01)
C07H 19/20 (2006.01)
European patent
(11) Number of the document 3661937
(13) Kind of document T
(96) European patent application number 18755368.0
Date of filing the European patent application 2018-07-30
(97) Date of publication of the European application 2020-06-10
(45) Date of publication and mention of the grant of the patent 2021-07-28
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2018/044415
Date 2018-07-30
PCT application publication
(87) Number WO 2019/027920
Date 2019-02-07
Priority applications
(30) Number Date Country code
201762539822 P 2017-08-01 US
Inventors
(72)
LAPINA, Olga Viktorovna , US
SHI, Bing , US
WANG, Silas , US
Grantee
(73) Gilead Sciences, Inc. , 333 Lakeside Drive, Foster City, CA 94404, US
Title
(54) CRYSTALLINE FORMS OF ETHYL ((S)-((((2R,5R)-5-(6-AMINO-9H-PURIN-9-YL)-4-FLUORO-2,5-DIHYDROFURAN-2-YL)OXY)METHYL)(PHENOXY)PHOSPHORYL)-L-ALANINATE (GS-9131) FOR TREATING VIRAL INFECTIONS
  CRYSTALLINE FORMS OF ETHYL ((S)-((((2R,5R)-5-(6-AMINO-9H-PURIN-9-YL)-4-FLUORO-2,5-DIHYDROFURAN-2-YL)OXY)METHYL)(PHENOXY)PHOSPHORYL)-L-ALANINATE (GS-9131) FOR TREATING VIRAL INFECTIONS