LT - PREPARATION PROCESS OF A CRYSTALLINE FORM OF 1-((2R,4R)-2-(1H-BENZO[D]IMIDAZOL-2-YL)-1-METHYLPIPERIDIN-4-YL)-3-(4-CYANOPHENYL)UREA MALEATE; A CRYSTALLINE FORM OF 1-((2R,4R)-2-(1H-BENZO[D]IMIDAZOL-2-YL)-1-METHYLPIPERIDIN-4-YL)-3-(4-CYANOPHENYL)UREA IMIDAZOLE COMPLEX (1:1)
EN - PREPARATION PROCESS OF A CRYSTALLINE FORM OF 1-((2R,4R)-2-(1H-BENZO[D]IMIDAZOL-2-YL)-1-METHYLPIPERIDIN-4-YL)-3-(4-CYANOPHENYL)UREA MALEATE; A CRYSTALLINE FORM OF 1-((2R,4R)-2-(1H-BENZO[D]IMIDAZOL-2-YL)-1-METHYLPIPERIDIN-4-YL)-3-(4-CYANOPHENYL)UREA IMIDAZOLE COMPLEX (1:1)
Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
| (51) |
INT.CL. |
C07D 401/04 |
(2006.01) |
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C07D 401/04 |
(2013.01) |
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A61P 35/00 |
(2006.01) |
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A61P 35/00 |
(2018.01) |
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A61P 43/00 |
(2006.01) |
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A61P 35/02 |
(2018.01) |
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A61P 43/00 |
(2018.01) |
Europos patentas
| (11) |
Patento numeris |
3666768 |
| (13) |
Dokumento rūšis |
T |
| (96) |
Europos patento paraiškos numeris |
20151107.8 |
|
Europos patento paraiškos padavimo data |
2016-04-13 |
| (97) |
Europos patento paraiškos paskelbimo data |
2020-06-17 |
| (45) |
Paskelbimo apie Europos patento išdavimą data |
2022-06-15
|
| (46) |
Apibrėžties vertimo paskelbimo data |
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Prioriteto paraiškos
| (30) |
Numeris |
Data |
Šalis |
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201562152108 P |
2015-04-24
|
US |
Išradėjai
| (72) |
HANSEN, Eric Christian , US
SEADEEK, Christopher Scott , US
RANE, Anil Mahadeo , US
|
Savininkas
| (73) |
Pfizer Inc. ,
235 East 42nd Street, New York, NY 10017,
US
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Pavadinimas
| (54) |
PREPARATION PROCESS OF A CRYSTALLINE FORM OF 1-((2R,4R)-2-(1H-BENZO[D]IMIDAZOL-2-YL)-1-METHYLPIPERIDIN-4-YL)-3-(4-CYANOPHENYL)UREA MALEATE; A CRYSTALLINE FORM OF 1-((2R,4R)-2-(1H-BENZO[D]IMIDAZOL-2-YL)-1-METHYLPIPERIDIN-4-YL)-3-(4-CYANOPHENYL)UREA IMIDAZOLE COMPLEX (1:1) |
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PREPARATION PROCESS OF A CRYSTALLINE FORM OF 1-((2R,4R)-2-(1H-BENZO[D]IMIDAZOL-2-YL)-1-METHYLPIPERIDIN-4-YL)-3-(4-CYANOPHENYL)UREA MALEATE; A CRYSTALLINE FORM OF 1-((2R,4R)-2-(1H-BENZO[D]IMIDAZOL-2-YL)-1-METHYLPIPERIDIN-4-YL)-3-(4-CYANOPHENYL)UREA IMIDAZOLE COMPLEX (1:1) |