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LT - MACROCYCLIZATION REACTIONS AND INTERMEDIATES USEFUL IN THE SYNTHESIS OF ANALOGS OF HALICHONDRIN B
EN - MACROCYCLIZATION REACTIONS AND INTERMEDIATES USEFUL IN THE SYNTHESIS OF ANALOGS OF HALICHONDRIN B

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 493/22 (2006.01)
C07D 307/28 (2013.01)
C07D 307/28 (2006.01)
C07D 407/06 (2013.01)
C07C 6/02 (2006.01)
C07F 9/6561 (2013.01)
C07F 9/40 (2006.01)
C07D 407/14 (2013.01)
C07F 7/1804 (2013.01)
C07D 493/22 (2013.01)
C07F 9/65586 (2013.01)
C07D 493/14 (2013.01)
European patent
(11) Number of the document 3689881
(13) Kind of document T
(96) European patent application number 20156829.2
Date of filing the European patent application 2014-11-04
(97) Date of publication of the European application 2020-08-05
(45) Date of publication and mention of the grant of the patent 2022-01-12
(46) Date of publication of the claims translation
Priority applications
(30) Number Date Country code
201361899697 P 2013-11-04 US
Inventors
(72)
FANG, Francis G , US
KIM, Dae-Shik , US
CHOI, Hyeong-Wook , US
CHASE, Charles E. , US
LEE, Jaemoon , US
Grantee
(73) Eisai R&D Management Co., Ltd. , 6-10, Koishikawa 4-chome, Bunkyo-ku, Tokyo 112-8088, JP
Title
(54) MACROCYCLIZATION REACTIONS AND INTERMEDIATES USEFUL IN THE SYNTHESIS OF ANALOGS OF HALICHONDRIN B
  MACROCYCLIZATION REACTIONS AND INTERMEDIATES USEFUL IN THE SYNTHESIS OF ANALOGS OF HALICHONDRIN B