LT - CRYSTALLINE 2-AMINO-2-(HYDROXYMETHYL)PROPANE-1,3-DIOL SALT OF 4-(4-(1-ISOPROPYL-7-OXO-1,4,6,7-TETRAHYDROSPIRO[INDAZOLE-5,4'-PIPERIDINE]-1'-CARBONYL)-6-METHOXYPYRIDIN-2-YL)BENZOIC ACID
EN - CRYSTALLINE 2-AMINO-2-(HYDROXYMETHYL)PROPANE-1,3-DIOL SALT OF 4-(4-(1-ISOPROPYL-7-OXO-1,4,6,7-TETRAHYDROSPIRO[INDAZOLE-5,4'-PIPERIDINE]-1'-CARBONYL)-6-METHOXYPYRIDIN-2-YL)BENZOIC ACID
Legal status
Patent not validated
Bibliographic data
Indications of the International Patent Classification (IPC)
| (51) |
INT.CL. |
C07D 471/10 |
(2006.01) |
|
|
C07C 215/10 |
(2013.01) |
|
|
C07C 215/10 |
(2006.01) |
|
|
C07D 471/10 |
(2013.01) |
|
|
A61P 1/16 |
(2006.01) |
|
|
A61P 1/16 |
(2018.01) |
|
|
A61P 3/10 |
(2006.01) |
|
|
A61P 3/10 |
(2018.01) |
|
|
A61K 31/438 |
(2006.01) |
European patent
| (11) |
Number of the document |
3713942 |
| (13) |
Kind of document |
T |
| (96) |
European patent application number |
18811658.6 |
|
Date of filing the European patent application |
2018-11-14 |
| (97) |
Date of publication of the European application |
2020-09-30 |
| (45) |
Date of publication and mention of the grant of the patent |
2023-03-08
|
| (46) |
Date of publication of the claims translation |
|
PCT application
| (86) |
Number |
PCT/IB2018/058966 |
|
Date |
2018-11-14 |
PCT application publication
| (87) |
Number |
WO 2019/102311 |
|
Date |
2019-05-31 |
Priority applications
| (30) |
Number |
Date |
Country code |
|
201762589256 P |
2017-11-21
|
US |
Inventors
| (72) |
FERNANDO, Dilinie , US
LACASSE, Shawn M. , US
WIGLESWORTH, Kristin , US
|
Grantee
| (73) |
Pfizer Inc. ,
66 Hudson Boulevard East, New York, NY 10001-2192,
US
|
Title
| (54) |
CRYSTALLINE 2-AMINO-2-(HYDROXYMETHYL)PROPANE-1,3-DIOL SALT OF 4-(4-(1-ISOPROPYL-7-OXO-1,4,6,7-TETRAHYDROSPIRO[INDAZOLE-5,4'-PIPERIDINE]-1'-CARBONYL)-6-METHOXYPYRIDIN-2-YL)BENZOIC ACID |
| |
CRYSTALLINE 2-AMINO-2-(HYDROXYMETHYL)PROPANE-1,3-DIOL SALT OF 4-(4-(1-ISOPROPYL-7-OXO-1,4,6,7-TETRAHYDROSPIRO[INDAZOLE-5,4'-PIPERIDINE]-1'-CARBONYL)-6-METHOXYPYRIDIN-2-YL)BENZOIC ACID |