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LT - CRYSTALLINE 2-AMINO-2-(HYDROXYMETHYL)PROPANE-1,3-DIOL SALT OF 4-(4-(1-ISOPROPYL-7-OXO-1,4,6,7-TETRAHYDROSPIRO[INDAZOLE-5,4'-PIPERIDINE]-1'-CARBONYL)-6-METHOXYPYRIDIN-2-YL)BENZOIC ACID
EN - CRYSTALLINE 2-AMINO-2-(HYDROXYMETHYL)PROPANE-1,3-DIOL SALT OF 4-(4-(1-ISOPROPYL-7-OXO-1,4,6,7-TETRAHYDROSPIRO[INDAZOLE-5,4'-PIPERIDINE]-1'-CARBONYL)-6-METHOXYPYRIDIN-2-YL)BENZOIC ACID

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 471/10 (2006.01)
C07C 215/10 (2013.01)
C07C 215/10 (2006.01)
C07D 471/10 (2013.01)
A61P 1/16 (2006.01)
A61P 1/16 (2018.01)
A61P 3/10 (2006.01)
A61P 3/10 (2018.01)
A61K 31/438 (2006.01)
European patent
(11) Number of the document 3713942
(13) Kind of document T
(96) European patent application number 18811658.6
Date of filing the European patent application 2018-11-14
(97) Date of publication of the European application 2020-09-30
(45) Date of publication and mention of the grant of the patent 2023-03-08
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/IB2018/058966
Date 2018-11-14
PCT application publication
(87) Number WO 2019/102311
Date 2019-05-31
Priority applications
(30) Number Date Country code
201762589256 P 2017-11-21 US
Inventors
(72)
FERNANDO, Dilinie , US
LACASSE, Shawn M. , US
WIGLESWORTH, Kristin , US
Grantee
(73) Pfizer Inc. , 66 Hudson Boulevard East, New York, NY 10001-2192, US
Title
(54) CRYSTALLINE 2-AMINO-2-(HYDROXYMETHYL)PROPANE-1,3-DIOL SALT OF 4-(4-(1-ISOPROPYL-7-OXO-1,4,6,7-TETRAHYDROSPIRO[INDAZOLE-5,4'-PIPERIDINE]-1'-CARBONYL)-6-METHOXYPYRIDIN-2-YL)BENZOIC ACID
  CRYSTALLINE 2-AMINO-2-(HYDROXYMETHYL)PROPANE-1,3-DIOL SALT OF 4-(4-(1-ISOPROPYL-7-OXO-1,4,6,7-TETRAHYDROSPIRO[INDAZOLE-5,4'-PIPERIDINE]-1'-CARBONYL)-6-METHOXYPYRIDIN-2-YL)BENZOIC ACID