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LT - PROCESS FOR PREPARING HALICHONDRIN MACROLIDES AND ANALOGS THEREOF BY A PRINS REACTION, AND INTERMEDIATES OF THIS PROCESS
EN - PROCESS FOR PREPARING HALICHONDRIN MACROLIDES AND ANALOGS THEREOF BY A PRINS REACTION, AND INTERMEDIATES OF THIS PROCESS

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 307/28 (2006.01)
C07D 407/06 (2013.01)
C07D 307/20 (2006.01)
C07D 407/14 (2013.01)
C07D 407/14 (2006.01)
C07D 493/04 (2013.01)
C07D 407/06 (2006.01)
C07D 493/22 (2013.01)
C07D 493/22 (2006.01)
C07D 307/20 (2013.01)
C07D 493/04 (2006.01)
C07D 307/28 (2013.01)
C07F 9/6561 (2006.01)
C07F 9/6561 (2013.01)
A61P 35/00 (2006.01)
A61P 35/00 (2018.01)
European patent
(11) Number of the document 3737673
(13) Kind of document T
(96) European patent application number 19735901.1
Date of filing the European patent application 2019-01-03
(97) Date of publication of the European application 2020-11-18
(45) Date of publication and mention of the grant of the patent 2024-03-06
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2019/012178
Date 2019-01-03
PCT application publication
(87) Number WO 2019/136145
Date 2019-07-11
Priority applications
(30) Number Date Country code
201862613307 P 2018-01-03 US
Inventors
(72)
CHOI, Hyeong-Wook , US
FANG, Francis G. , US
Grantee
(73) Eisai R&D Management Co., Ltd. , 6-10 Koishikawa, 4-Chome Bunkyo-Ku, Tokyo 112-8088, JP
Title
(54) PROCESS FOR PREPARING HALICHONDRIN MACROLIDES AND ANALOGS THEREOF BY A PRINS REACTION, AND INTERMEDIATES OF THIS PROCESS
  PROCESS FOR PREPARING HALICHONDRIN MACROLIDES AND ANALOGS THEREOF BY A PRINS REACTION, AND INTERMEDIATES OF THIS PROCESS