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LT - TRICYCLIC HETEROCYCLE COMPOUNDS USEFUL AS HIV INTEGRASE INHIBITORS
EN - TRICYCLIC HETEROCYCLE COMPOUNDS USEFUL AS HIV INTEGRASE INHIBITORS

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Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 471/08 (2006.01)
A61K 45/06 (2013.01)
C07D 471/18 (2006.01)
C07D 498/18 (2013.01)
C07D 498/18 (2006.01)
C07D 471/18 (2013.01)
A61K 31/395 (2006.01)
C07D 471/08 (2013.01)
A61K 31/53 (2006.01)
A61P 31/18 (2018.01)
A61K 31/5365 (2006.01)
C07D 471/02 (2006.01)
C07D 471/12 (2006.01)
C07D 471/16 (2006.01)
A61P 31/18 (2006.01)
European patent
(11) Number of the document 3752144
(13) Kind of document T
(96) European patent application number 19754182.4
Date of filing the European patent application 2019-02-11
(97) Date of publication of the European application 2020-12-23
(45) Date of publication and mention of the grant of the patent 2022-12-28
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2019/017409
Date 2019-02-11
PCT application publication
(87) Number WO 2019/160783
Date 2019-08-22
Priority applications
(30) Number Date Country code
201862630974 P 2018-02-15 US
Inventors
(72)
EMBREY, Mark, W. , US
HARTINGH, Timothy John , US
LABROLI, Marc , US
RAHEEM, Izzat, T. , US
Grantee
(73) Merck Sharp & Dohme LLC , 126 East Lincoln Avenue, Rahway, New Jersey 07065, US
Title
(54) TRICYCLIC HETEROCYCLE COMPOUNDS USEFUL AS HIV INTEGRASE INHIBITORS
  TRICYCLIC HETEROCYCLE COMPOUNDS USEFUL AS HIV INTEGRASE INHIBITORS