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Patent in force
(51) | INT.CL. | A61P 35/00 | (2006.01) |
C07D 471/04 | (2006.01) | ||
A61K 31/437 | (2006.01) |
(11) | Number of the document | 3810283 |
(13) | Kind of document | T |
(96) | European patent application number | 19745335.0 |
Date of filing the European patent application | 2019-06-17 | |
(97) | Date of publication of the European application | 2021-04-28 |
(45) | Date of publication and mention of the grant of the patent | 2023-06-14 |
(46) | Date of publication of the claims translation | 2023-08-25 |
(86) | Number | PCT/US2019/037492 |
Date | 2019-06-17 |
(87) | Number | WO 2019/245974 |
Date | 2019-12-26 |
(30) | Number | Date | Country code |
201862687930 P | 2018-06-21 | US | |
201862719896 P | 2018-08-20 | US |
(72) |
CHUNG, Cheol Keun , US
XU, Jie , US
IDING, Hans , CH
CLAGG, Kyle , US
DALZIEL, Michael , US
FETTES, Alec , CH
GOSSELIN, Francis , US
LIM, Ngiap-Kie , US
MCCLORY, Andrew , US
ZHANG, Haiming , US
CHAKRAVARTY, Paroma , US
NAGAPUDI, Kartik , US
ROBINSON, Sarah , US
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(73) |
F. Hoffmann-La Roche AG ,
Grenzacherstrasse 124, 4070 Basel,
CH
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(74) |
Reda ŽABOLIENĖ,
METIDA, Verslo centras "VERTAS", Gynėjų g. 16, LT-01109 Vilnius,
LT
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(54) | 3-((1R,3R)-1-(2,6-difluor-4-((1-(3-fluorpropil)azetidin-3- il)amino) fenil)-3-metil-1,3,4,9-tetrahidro-2H-pirido[3,4-b]indol-2-il)- 2,2- difluorpropan-1-olio tartrato druskos kietosios formos, jų paruošimo procesas ir jų naudojimo būdai vėžiui gydyti |
SOLID FORMS OF THE TARTRATE SALT OF 3-((1R,3R)-1-(2,6-DIFLUORO-4-((1-(3-FLUOROPROPYL)AZETIDIN-3-YL)AMINO)PHENYL)-3-METHYL-1,3,4,9-TETRAHYDRO-2H-PYRIDO[3,4-B]INDOL-2-YL)-2,2-DIFLUOROPROPAN-1-OL, PROCESS FOR THEIR PREPARATION AND METHODS OF THEIR USE IN TREATING CANCERS |
Payment date | Validity (years) | Amount | |
2025-05-20 | 7 | 162.00 EUR |
2026-06-17 |