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LT - 3-((1R,3R)-1-(2,6-difluor-4-((1-(3-fluorpropil)azetidin-3- il)amino) fenil)-3-metil-1,3,4,9-tetrahidro-2H-pirido[3,4-b]indol-2-il)- 2,2- difluorpropan-1-olio tartrato druskos kietosios formos, jų paruošimo procesas ir jų naudojimo būdai vėžiui gydyti
EN - SOLID FORMS OF THE TARTRATE SALT OF 3-((1R,3R)-1-(2,6-DIFLUORO-4-((1-(3-FLUOROPROPYL)AZETIDIN-3-YL)AMINO)PHENYL)-3-METHYL-1,3,4,9-TETRAHYDRO-2H-PYRIDO[3,4-B]INDOL-2-YL)-2,2-DIFLUOROPROPAN-1-OL, PROCESS FOR THEIR PREPARATION AND METHODS OF THEIR USE IN TREATING CANCERS

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Patent in force

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. A61P 35/00 (2006.01)
C07D 471/04 (2006.01)
A61K 31/437 (2006.01)
European patent
(11) Number of the document 3810283
(13) Kind of document T
(96) European patent application number 19745335.0
Date of filing the European patent application 2019-06-17
(97) Date of publication of the European application 2021-04-28
(45) Date of publication and mention of the grant of the patent 2023-06-14
(46) Date of publication of the claims translation 2023-08-25
PCT application
(86) Number PCT/US2019/037492
Date 2019-06-17
PCT application publication
(87) Number WO 2019/245974
Date 2019-12-26
Priority applications
(30) Number Date Country code
201862687930 P 2018-06-21 US
201862719896 P 2018-08-20 US
Inventors
(72)
CHUNG, Cheol Keun , US
XU, Jie , US
IDING, Hans , CH
CLAGG, Kyle , US
DALZIEL, Michael , US
FETTES, Alec , CH
GOSSELIN, Francis , US
LIM, Ngiap-Kie , US
MCCLORY, Andrew , US
ZHANG, Haiming , US
CHAKRAVARTY, Paroma , US
NAGAPUDI, Kartik , US
ROBINSON, Sarah , US
Grantee
(73) F. Hoffmann-La Roche AG , Grenzacherstrasse 124, 4070 Basel, CH
Attorney or representative
(74) Reda ŽABOLIENĖ, METIDA, Verslo centras "VERTAS", Gynėjų g. 16, LT-01109 Vilnius, LT
Title
(54) 3-((1R,3R)-1-(2,6-difluor-4-((1-(3-fluorpropil)azetidin-3- il)amino) fenil)-3-metil-1,3,4,9-tetrahidro-2H-pirido[3,4-b]indol-2-il)- 2,2- difluorpropan-1-olio tartrato druskos kietosios formos, jų paruošimo procesas ir jų naudojimo būdai vėžiui gydyti
  SOLID FORMS OF THE TARTRATE SALT OF 3-((1R,3R)-1-(2,6-DIFLUORO-4-((1-(3-FLUOROPROPYL)AZETIDIN-3-YL)AMINO)PHENYL)-3-METHYL-1,3,4,9-TETRAHYDRO-2H-PYRIDO[3,4-B]INDOL-2-YL)-2,2-DIFLUOROPROPAN-1-OL, PROCESS FOR THEIR PREPARATION AND METHODS OF THEIR USE IN TREATING CANCERS
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2026-06-17