LT - PROCESS FOR THE PREPARATION OF METHYL 6-(2,4-DICHLOROPHENYL)-5-[4-[(3S)-1-(3-FLUOROPROPYL)PYRROLIDIN-3-YL]OXYPHENYL]-8,9-DIHYDRO-7H-BENZO[7]ANNULENE-2-CARBOXYLATE AND A SALT THEREOF
EN - PROCESS FOR THE PREPARATION OF METHYL 6-(2,4-DICHLOROPHENYL)-5-[4-[(3S)-1-(3-FLUOROPROPYL)PYRROLIDIN-3-YL]OXYPHENYL]-8,9-DIHYDRO-7H-BENZO[7]ANNULENE-2-CARBOXYLATE AND A SALT THEREOF
Legal status
Patent not validated
Bibliographic data
Indications of the International Patent Classification (IPC)
(51) |
INT.CL. |
C07D 207/12 |
(2006.01) |
|
|
C07D 207/12 |
(2013.01) |
|
|
C07C 59/255 |
(2013.01) |
|
|
C07C 55/07 |
(2013.01) |
European patent
(11) |
Number of the document |
3847157 |
(13) |
Kind of document |
T |
(96) |
European patent application number |
19765711.7 |
|
Date of filing the European patent application |
2019-09-06 |
(97) |
Date of publication of the European application |
2021-07-14 |
(45) |
Date of publication and mention of the grant of the patent |
2022-05-18
|
(46) |
Date of publication of the claims translation |
|
PCT application
(86) |
Number |
PCT/EP2019/073827 |
|
Date |
2019-09-06 |
PCT application publication
(87) |
Number |
WO 2020/049153 |
|
Date |
2020-03-12 |
Priority applications
(30) |
Number |
Date |
Country code |
|
18306177 |
2018-09-07
|
EP |
Inventors
(72) |
RABION, Alain , FR
TABART, Michel , FR
WEHREY, Christian , FR
|
Grantee
(73) |
SANOFI ,
54 rue La Boétie, 75008 Paris,
FR
|
Title
(54) |
PROCESS FOR THE PREPARATION OF METHYL 6-(2,4-DICHLOROPHENYL)-5-[4-[(3S)-1-(3-FLUOROPROPYL)PYRROLIDIN-3-YL]OXYPHENYL]-8,9-DIHYDRO-7H-BENZO[7]ANNULENE-2-CARBOXYLATE AND A SALT THEREOF |
|
PROCESS FOR THE PREPARATION OF METHYL 6-(2,4-DICHLOROPHENYL)-5-[4-[(3S)-1-(3-FLUOROPROPYL)PYRROLIDIN-3-YL]OXYPHENYL]-8,9-DIHYDRO-7H-BENZO[7]ANNULENE-2-CARBOXYLATE AND A SALT THEREOF |