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LT - PROCESS FOR THE PREPARATION OF METHYL 6-(2,4-DICHLOROPHENYL)-5-[4-[(3S)-1-(3-FLUOROPROPYL)PYRROLIDIN-3-YL]OXYPHENYL]-8,9-DIHYDRO-7H-BENZO[7]ANNULENE-2-CARBOXYLATE AND A SALT THEREOF
EN - PROCESS FOR THE PREPARATION OF METHYL 6-(2,4-DICHLOROPHENYL)-5-[4-[(3S)-1-(3-FLUOROPROPYL)PYRROLIDIN-3-YL]OXYPHENYL]-8,9-DIHYDRO-7H-BENZO[7]ANNULENE-2-CARBOXYLATE AND A SALT THEREOF

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 207/12 (2006.01)
C07D 207/12 (2013.01)
C07C 59/255 (2013.01)
C07C 55/07 (2013.01)
European patent
(11) Number of the document 3847157
(13) Kind of document T
(96) European patent application number 19765711.7
Date of filing the European patent application 2019-09-06
(97) Date of publication of the European application 2021-07-14
(45) Date of publication and mention of the grant of the patent 2022-05-18
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/EP2019/073827
Date 2019-09-06
PCT application publication
(87) Number WO 2020/049153
Date 2020-03-12
Priority applications
(30) Number Date Country code
18306177 2018-09-07 EP
Inventors
(72)
RABION, Alain , FR
TABART, Michel , FR
WEHREY, Christian , FR
Grantee
(73) SANOFI , 54 rue La Boétie, 75008 Paris, FR
Title
(54) PROCESS FOR THE PREPARATION OF METHYL 6-(2,4-DICHLOROPHENYL)-5-[4-[(3S)-1-(3-FLUOROPROPYL)PYRROLIDIN-3-YL]OXYPHENYL]-8,9-DIHYDRO-7H-BENZO[7]ANNULENE-2-CARBOXYLATE AND A SALT THEREOF
  PROCESS FOR THE PREPARATION OF METHYL 6-(2,4-DICHLOROPHENYL)-5-[4-[(3S)-1-(3-FLUOROPROPYL)PYRROLIDIN-3-YL]OXYPHENYL]-8,9-DIHYDRO-7H-BENZO[7]ANNULENE-2-CARBOXYLATE AND A SALT THEREOF