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LT - 11-HYDROXYL-6-SUBSTITUTED-DERIVATIVES OF BILE ACIDS AND AMINO ACID CONJUGATES THEREOF AS FARNESOID X RECEPTOR MODULATORS
EN - 11-HYDROXYL-6-SUBSTITUTED-DERIVATIVES OF BILE ACIDS AND AMINO ACID CONJUGATES THEREOF AS FARNESOID X RECEPTOR MODULATORS

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. A61K 31/575 (2006.01)
C07J 31/006 (2013.01)
C07J 9/00 (2006.01)
C07J 41/0061 (2013.01)
C07J 41/00 (2006.01)
C07J 71/001 (2013.01)
A61P 1/16 (2006.01)
A61P 1/16 (2018.01)
A61P 11/00 (2006.01)
A61P 1/00 (2018.01)
A61P 13/00 (2006.01)
C07J 9/005 (2013.01)
A61P 43/00 (2006.01)
A61K 31/575 (2013.01)
A61P 1/00 (2006.01)
A61P 43/00 (2018.01)
C07J 71/00 (2006.01)
A61P 11/00 (2018.01)
C07J 31/00 (2006.01)
A61P 13/00 (2018.01)
European patent
(11) Number of the document 3848038
(13) Kind of document T
(96) European patent application number 20211780.0
Date of filing the European patent application 2014-05-14
(97) Date of publication of the European application 2021-07-14
(45) Date of publication and mention of the grant of the patent 2022-11-09
(46) Date of publication of the claims translation
Priority applications
(30) Number Date Country code
201361823169 P 2013-05-14 US
Inventors
(72)
PELLICCIARI, Roberto , IT
Grantee
(73) Intercept Pharmaceuticals, Inc. , 305 Madison Avenue, Morristown NJ 07960, US
Title
(54) 11-HYDROXYL-6-SUBSTITUTED-DERIVATIVES OF BILE ACIDS AND AMINO ACID CONJUGATES THEREOF AS FARNESOID X RECEPTOR MODULATORS
  11-HYDROXYL-6-SUBSTITUTED-DERIVATIVES OF BILE ACIDS AND AMINO ACID CONJUGATES THEREOF AS FARNESOID X RECEPTOR MODULATORS