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LT - PYRIMIDONE DERIVATIVES AS SELECTIVE CYTOTOXIC AGENTS AGAINST HIV INFECTED CELLS
EN - PYRIMIDONE DERIVATIVES AS SELECTIVE CYTOTOXIC AGENTS AGAINST HIV INFECTED CELLS

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Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 239/52 (2006.01)
C07D 239/52 (2013.01)
A61K 31/505 (2006.01)
A61P 31/18 (2018.01)
A61P 31/18 (2006.01)
European patent
(11) Number of the document 3898595
(13) Kind of document T
(96) European patent application number 19845846.5
Date of filing the European patent application 2019-12-13
(97) Date of publication of the European application 2021-10-27
(45) Date of publication and mention of the grant of the patent 2024-05-01
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2019/066125
Date 2019-12-13
PCT application publication
(87) Number WO 2020/131597
Date 2020-06-25
Priority applications
(30) Number Date Country code
201862781356 P 2018-12-18 US
Inventors
(72)
CONVERSO, Antonella , US
EL MARROUNI, Abdellatif , US
FORSTER, Ashley , US
FRIE, Jessica, L. , US
HUNTER, David, N. , US
KUDUK, Scott, D. , US
MITCHELL, Helen, J. , US
NANTERMET, Philippe , US
SHA, Deyou , US
SHIPE, William Daniel , US
WANG, Cheng , US
WANG, Deping , US
Grantee
(73) Merck Sharp & Dohme LLC , 126 East Lincoln Avenue, Rahway, New Jersey 07065, US
Title
(54) PYRIMIDONE DERIVATIVES AS SELECTIVE CYTOTOXIC AGENTS AGAINST HIV INFECTED CELLS
  PYRIMIDONE DERIVATIVES AS SELECTIVE CYTOTOXIC AGENTS AGAINST HIV INFECTED CELLS