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LT - 1H-INDAZOLE-3-CARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS FACTOR D INHIBITORS FOR TREATING DISEASES CHARACTERIZED BY ABERRANT COMPLEMENT SYSTEM ACTIVITY, SUCH AS E.G. IMMUNOLOGICAL DISORDERS
EN - 1H-INDAZOLE-3-CARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS FACTOR D INHIBITORS FOR TREATING DISEASES CHARACTERIZED BY ABERRANT COMPLEMENT SYSTEM ACTIVITY, SUCH AS E.G. IMMUNOLOGICAL DISORDERS

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 403/12 (2013.01)
C07D 401/12 (2006.01)
C07D 231/56 (2006.01)
C07D 401/14 (2013.01)
C07D 231/56 (2013.01)
C07D 209/40 (2006.01)
C07D 401/04 (2013.01)
C07D 209/48 (2006.01)
C07D 401/06 (2013.01)
C07D 487/04 (2006.01)
C07D 471/04 (2006.01)
C07D 401/12 (2013.01)
C07D 403/12 (2006.01)
C07D 403/04 (2013.01)
C07D 403/04 (2006.01)
C07D 403/06 (2013.01)
C07D 403/06 (2006.01)
C07D 405/12 (2013.01)
C07D 471/04 (2013.01)
C07D 401/14 (2006.01)
C07D 487/04 (2013.01)
C07D 401/04 (2006.01)
C07D 401/06 (2006.01)
C07D 209/12 (2013.01)
C07D 405/12 (2006.01)
C07D 209/40 (2013.01)
C07D 209/12 (2006.01)
C07D 209/42 (2013.01)
C07D 209/48 (2013.01)
C07D 209/42 (2006.01)
A61P 21/04 (2018.01)
A61K 31/416 (2006.01)
A61P 25/28 (2018.01)
A61P 37/00 (2006.01)
A61P 9/00 (2018.01)
A61P 37/06 (2006.01)
A61P 37/06 (2018.01)
A61P 25/00 (2006.01)
A61P 13/00 (2018.01)
A61P 21/04 (2006.01)
A61K 31/416 (2013.01)
A61K 31/4439 (2006.01)
Y02A 50/30 (2018.01)
A61K 31/404 (2006.01)
A61P 13/00 (2006.01)
A61K 31/4035 (2006.01)
A61P 13/12 (2006.01)
A61P 25/28 (2006.01)
A61P 9/00 (2006.01)
European patent
(11) Number of the document 3925956
(13) Kind of document T
(96) European patent application number 21173901.6
Date of filing the European patent application 2017-02-01
(97) Date of publication of the European application 2021-12-22
(45) Date of publication and mention of the grant of the patent 2024-04-10
(46) Date of publication of the claims translation
Priority applications
(30) Number Date Country code
201662289653 P 2016-02-01 US
Inventors
(72)
KOTIAN, Pravin, L , US
BABU, Yarlagadda, S. , US
ZHANG, Weihe , US
VOGETI, Lakshminarayana , US
WU, Minwan , US
CHINTAREDDY, Venkat, R. , US
RAMAN, Krishnan , US
Grantee
(73) BioCryst Pharmaceuticals, Inc. , 4505 Emperor Blvd., Durham, NC 27703, US
Title
(54) 1H-INDAZOLE-3-CARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS FACTOR D INHIBITORS FOR TREATING DISEASES CHARACTERIZED BY ABERRANT COMPLEMENT SYSTEM ACTIVITY, SUCH AS E.G. IMMUNOLOGICAL DISORDERS
  1H-INDAZOLE-3-CARBOXAMIDE DERIVATIVES AND RELATED COMPOUNDS AS FACTOR D INHIBITORS FOR TREATING DISEASES CHARACTERIZED BY ABERRANT COMPLEMENT SYSTEM ACTIVITY, SUCH AS E.G. IMMUNOLOGICAL DISORDERS