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LT - PROCESSES FOR PREPARING (3R,4R)-1-BENZYL-N,4-DIMETHYLPIPERIDIN-3-AMINE OR A SALT THEREOF AND PROCESSES FOR PREPARING TOFACITINIB USING THE SAME
EN - PROCESSES FOR PREPARING (3R,4R)-1-BENZYL-N,4-DIMETHYLPIPERIDIN-3-AMINE OR A SALT THEREOF AND PROCESSES FOR PREPARING TOFACITINIB USING THE SAME

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 211/56 (2006.01)
A61P 1/00 (2018.01)
C07D 211/02 (2006.01)
A61P 19/02 (2018.01)
A61P 1/00 (2006.01)
A61P 29/00 (2018.01)
A61P 19/02 (2006.01)
C07D 211/02 (2013.01)
A61P 29/00 (2006.01)
C07D 211/56 (2013.01)
C07D 487/04 (2006.01)
C07D 487/04 (2013.01)
European patent
(11) Number of the document 3927689
(13) Kind of document T
(96) European patent application number 20783663.6
Date of filing the European patent application 2020-04-03
(97) Date of publication of the European application 2021-12-29
(45) Date of publication and mention of the grant of the patent 2024-01-24
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/KR2020/004547
Date 2020-04-03
PCT application publication
(87) Number WO 2020/204647
Date 2020-10-08
Priority applications
(30) Number Date Country code
20190040383 2019-04-05 KR
Inventors
(72)
OH, Sang-Ho , KR
LEE, Doo-Byung , KR
KWON, Kyoung-Chan , KR
KIM, Sang-Won , KR
HWANG, Hyo-Ick , KR
LEE, Kyeong-Sill , KR
JO, Ik-Su , KR
CHOI, Ji-Hye , KR
CHO, Sung-Hee , KR
LEE, Su-Young , KR
Grantee
(73) Yuhan Corporation , 74 Noryangjin-ro Dongjak-gu, Seoul 06927, KR
Title
(54) PROCESSES FOR PREPARING (3R,4R)-1-BENZYL-N,4-DIMETHYLPIPERIDIN-3-AMINE OR A SALT THEREOF AND PROCESSES FOR PREPARING TOFACITINIB USING THE SAME
  PROCESSES FOR PREPARING (3R,4R)-1-BENZYL-N,4-DIMETHYLPIPERIDIN-3-AMINE OR A SALT THEREOF AND PROCESSES FOR PREPARING TOFACITINIB USING THE SAME