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LT - (R)-3-(3-CHLORO-5-FLUORO-2-((4-(1H-PYRAZOL-1-YL)-2-METHYLQUINOLIN-8-YLOXY)METHYL)PHENYL)MORPHOLINE DERIVATIVES AND RELATED COMPOUNDS AS BRADYKININ (BK) B2 RECEPTOR ANTAGONIST FOR TREATING SKIN DISEASES
EN - (R)-3-(3-CHLORO-5-FLUORO-2-((4-(1H-PYRAZOL-1-YL)-2-METHYLQUINOLIN-8-YLOXY)METHYL)PHENYL)MORPHOLINE DERIVATIVES AND RELATED COMPOUNDS AS BRADYKININ (BK) B2 RECEPTOR ANTAGONIST FOR TREATING SKIN DISEASES

Teisinis statusas

Patentas galioja

Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) INT.CL. C07D 413/14 (2006.01)
A61K 31/4709 (2006.01)
A61K 31/5377 (2006.01)
A61K 31/4155 (2006.01)
A61K 31/4196 (2006.01)
A61K 31/422 (2006.01)
A61P 1/16 (2006.01)
A61P 5/00 (2006.01)
A61P 9/00 (2006.01)
A61P 11/00 (2006.01)
A61P 13/00 (2006.01)
A61P 13/12 (2006.01)
A61P 15/00 (2006.01)
A61P 17/00 (2006.01)
A61P 25/00 (2006.01)
Europos patentas
(11) Patento numeris 3956326
(13) Dokumento rūšis T
(96) Europos patento paraiškos numeris 20732117.5
Europos patento paraiškos padavimo data 2020-05-25
(97) Europos patento paraiškos paskelbimo data 2022-02-23
(45) Paskelbimo apie Europos patento išdavimą data 2023-06-28
(46) Apibrėžties vertimo paskelbimo data
Tarptautinės paraiškos padavimo
(86) Numeris PCT/EP2020/064379
Data 2020-05-25
Tarptautinės paraiškos paskelbimo
(87) Numeris WO 2020/234480
Data 2020-11-26
Prioriteto paraiškos
(30) Numeris Data Šalis
19176229 2019-05-23 EP
Išradėjai
(72)
GIBSON, Christoph , DE
SAUPE, Joern , DE
AMBROSI, Horst-Dieter , DE
HAUSTEDT, Lars Ole , DE
Savininkas
(73) Pharvaris GmbH , Grafenauweg 8, 6300 Zug, CH
Pavadinimas
(54) (R)-3-(3-CHLORO-5-FLUORO-2-((4-(1H-PYRAZOL-1-YL)-2-METHYLQUINOLIN-8-YLOXY)METHYL)PHENYL)MORPHOLINE DERIVATIVES AND RELATED COMPOUNDS AS BRADYKININ (BK) B2 RECEPTOR ANTAGONIST FOR TREATING SKIN DISEASES
  (R)-3-(3-CHLORO-5-FLUORO-2-((4-(1H-PYRAZOL-1-YL)-2-METHYLQUINOLIN-8-YLOXY)METHYL)PHENYL)MORPHOLINE DERIVATIVES AND RELATED COMPOUNDS AS BRADYKININ (BK) B2 RECEPTOR ANTAGONIST FOR TREATING SKIN DISEASES