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LT - COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF HIF2-ALPHA AND THEIR METHODS OF USE
EN - COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF HIF2-ALPHA AND THEIR METHODS OF USE

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Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 471/04 (2006.01)
A61P 35/00 (2018.01)
C07D 519/00 (2006.01)
C07D 471/04 (2013.01)
A61P 35/00 (2006.01)
C07D 519/00 (2013.01)
A61K 31/437 (2006.01)
A61K 45/06 (2013.01)
European patent
(11) Number of the document 4143187
(13) Kind of document T
(96) European patent application number 21723390.7
Date of filing the European patent application 2021-04-27
(97) Date of publication of the European application 2023-03-08
(45) Date of publication and mention of the grant of the patent 2024-05-08
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/IB2021/053486
Date 2021-04-27
PCT application publication
(87) Number WO 2021/220170
Date 2021-11-04
Priority applications
(30) Number Date Country code
PCT/CN2020/087831 2020-04-29 WO
Inventors
(72)
FAIRHURST, Robin Alec , CH
FRITSCH, Christine , CH
GERSPACHER, Marc , CH
HINRICHS, Jürgen Hans-Hermann , CH
LANGLOIS, Jean-Baptiste Georges Armand , CH
LEBLANC, Catherine , CH
LI, Tengfei , CN
LORTHIOIS, Edwige Liliane Jeanne , CH
MURA, Christophe , CH
NIETO-OBERHUBER, Cristina Montserrat , CH
TODOROV, Milen , CH
VAUPEL, Andrea , CH
WARIN, Nicolas , CH
WILCKEN, Rainer , CH
Grantee
(73) Novartis AG , Lichtstrasse 35, 4056 Basel, CH
Title
(54) COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF HIF2-ALPHA AND THEIR METHODS OF USE
  COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF HIF2-ALPHA AND THEIR METHODS OF USE