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Legal status
Patent not validated
| (51) | INT.CL. | C07D 471/04 | (2006.01) |
| A61P 35/00 | (2018.01) | ||
| C07D 519/00 | (2006.01) | ||
| C07D 471/04 | (2013.01) | ||
| A61P 35/00 | (2006.01) | ||
| C07D 519/00 | (2013.01) | ||
| A61K 31/437 | (2006.01) | ||
| A61K 45/06 | (2013.01) |
| (11) | Number of the document | 4143187 |
| (13) | Kind of document | T |
| (96) | European patent application number | 21723390.7 |
| Date of filing the European patent application | 2021-04-27 | |
| (97) | Date of publication of the European application | 2023-03-08 |
| (45) | Date of publication and mention of the grant of the patent | 2024-05-08 |
| (46) | Date of publication of the claims translation |
| (86) | Number | PCT/IB2021/053486 |
| Date | 2021-04-27 |
| (87) | Number | WO 2021/220170 |
| Date | 2021-11-04 |
| (30) | Number | Date | Country code |
| PCT/CN2020/087831 | 2020-04-29 | WO |
| (72) |
FAIRHURST, Robin Alec , CH
FRITSCH, Christine , CH
GERSPACHER, Marc , CH
HINRICHS, Jürgen Hans-Hermann , CH
LANGLOIS, Jean-Baptiste Georges Armand , CH
LEBLANC, Catherine , CH
LI, Tengfei , CN
LORTHIOIS, Edwige Liliane Jeanne , CH
MURA, Christophe , CH
NIETO-OBERHUBER, Cristina Montserrat , CH
TODOROV, Milen , CH
VAUPEL, Andrea , CH
WARIN, Nicolas , CH
WILCKEN, Rainer , CH
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| (73) |
Novartis AG ,
Lichtstrasse 35, 4056 Basel,
CH
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| (54) | COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF HIF2-ALPHA AND THEIR METHODS OF USE |
| COMPOUNDS AND COMPOSITIONS FOR INHIBITING THE ACTIVITY OF HIF2-ALPHA AND THEIR METHODS OF USE |