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LT - SUBSTITUTED PYRAZOLES AS HUMAN PLASMA KALLIKREIN INHIBITORS
EN - SUBSTITUTED PYRAZOLES AS HUMAN PLASMA KALLIKREIN INHIBITORS

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 403/04 (2006.01)
C07D 403/12 (2013.01)
C07D 403/14 (2006.01)
C07D 401/14 (2013.01)
A61P 1/02 (2006.01)
C07D 401/04 (2013.01)
C07D 231/14 (2006.01)
C07D 401/12 (2013.01)
A61P 1/04 (2006.01)
C07D 403/04 (2013.01)
A61P 3/10 (2006.01)
C07D 405/12 (2013.01)
C07D 413/04 (2013.01)
A61P 7/00 (2006.01)
A61P 9/00 (2006.01)
C07D 413/12 (2013.01)
C07D 417/12 (2013.01)
A61P 11/04 (2006.01)
C07D 231/14 (2013.01)
A61P 13/02 (2006.01)
A61P 1/02 (2018.01)
C07D 401/04 (2006.01)
A61P 1/04 (2018.01)
C07D 401/12 (2006.01)
A61P 11/04 (2018.01)
C07D 401/14 (2006.01)
A61P 13/02 (2018.01)
C07D 403/12 (2006.01)
A61P 13/12 (2018.01)
C07D 405/12 (2006.01)
C07D 413/12 (2006.01)
A61P 19/02 (2018.01)
A61P 25/00 (2018.01)
C07D 417/12 (2006.01)
A61P 27/02 (2018.01)
A61P 29/00 (2018.01)
A61P 31/04 (2018.01)
A61P 43/00 (2018.01)
A61P 7/00 (2018.01)
A61P 7/02 (2018.01)
A61P 7/04 (2018.01)
A61P 7/10 (2018.01)
A61P 9/00 (2018.01)
A61P 9/10 (2018.01)
A61P 9/12 (2018.01)
A61P 3/10 (2018.01)
C07D 403/14 (2013.01)
European patent
(11) Number of the document 4180424
(13) Kind of document T
(96) European patent application number 22191079.7
Date of filing the European patent application 2015-03-09
(97) Date of publication of the European application 2023-05-17
(45) Date of publication and mention of the grant of the patent 2025-06-25
(46) Date of publication of the claims translation
Priority applications
(30) Number Date Country code
201461949808 P 2014-03-07 US
201461981515 P 2014-04-18 US
Inventors
(72)
KOTIAN, Pravin L. , US
BABU, Yarlagadda S. , US
WU, Minwan , US
KUMAR, Satish V , US
ZHANG, Weihe , US
CHINTAREDDY, Venkat R , US
Grantee
(73) BioCryst Pharmaceuticals, Inc. , 4505 Emperor Blvd., Durham, NC 27703, US
Title
(54) SUBSTITUTED PYRAZOLES AS HUMAN PLASMA KALLIKREIN INHIBITORS
  SUBSTITUTED PYRAZOLES AS HUMAN PLASMA KALLIKREIN INHIBITORS