LT - (4R,5S,6S,7R)-heksahidro-1-[5-(3-aminoinazol)metil]-3-butil-5, 6-dihidroksi-4,7-bis[fenilmetil]-2H-1,3-diazepin-2-onas, jo gavimas ir jo kaip ŽIV proteazės inhibitoriaus panaudojimas
EN - (4R,5S,6S,7R)-HEXAHYDRO-1-[5-(3-AMINOINAZOLE)METHYL]-BUTYL-5,6-DIHYDROXY-4,7-BIS[PHENYLMETHYL]-2H-1,3-DIAZEPIN-2-ONE, ITS PREPARATION AND ITS USE AS HIV PROTEASE INHIBITOR
Legal status
Patent lapsed (non-payment of fees)
Bibliographic data
Indications of the International Patent Classification (IPC)
| (51) |
INT.CL.: (2006.01) |
A61K 31/33
A61K 31/55
C07D 243/00
C07D 403/00
|
Patent
| (11) |
Number of the document |
4619 |
| (13) |
Kind of document |
B |
| (21) |
Application number |
99-045 |
| (22) |
Date of filing the application |
1999-05-03 |
| (41) |
Date of publication of the application |
1999-09-27 |
| (45) |
Date of publication of patent |
2000-02-25 |
PCT application
| (86) |
Number |
PCT/US97/20036 |
|
Date |
1997-11-04 |
PCT application publication
| (87) |
Number |
WO 98/20009 |
|
Date |
1998-05-14 |
Priority applications
| (30) |
Number |
Date |
Country code |
|
747103 |
1996-11-08
|
US |
|
029746 |
1996-11-08
|
US |
Applicant
| (71) |
DUPONT PHARMACEUTICALS COMPANY,
Chestnut Run Plaza, 974 Centre Road, Wilmington, Delaware,
US
|
Inventors
| (72) |
James David RODGERS, US
Patrick Yuk-Sun LAM, US
|
Grantee
| (73) |
DUPONT PHARMACEUTICALS COMPANY,
Chestnut Run Plaza, 974 Centre Road, Wilmington, Delaware,
US
|
Attorney or representative
| (74) |
Reda ŽABOLIENĖ,
METIDA, Verslo centras "VERTAS", Gynėjų g. 16, LT-01109 Vilnius,
LT
|
Title
| (54) |
(4R,5S,6S,7R)-HEXAHYDRO-1-[5-(3-AMINOINAZOLE)METHYL]-BUTYL-5,6-DIHYDROXY-4,7-BIS[PHENYLMETHYL]-2H-1,3-DIAZEPIN-2-ONE, ITS PREPARATION AND ITS USE AS HIV PROTEASE INHIBITOR
|
Last renewal fee
|
Payment date |
Validity (years) |
Amount |
|
2001-10-05 |
5 |
400.00
LTL
|
Legal status
|
Patent lapsed (non-payment of fees)
|
|
|
Invalidation date |
2002-11-04 |
