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LT - PROCESS FOR THE MANUFACTURE OF THE CALCIUM SALT OF ROSUVASTATIN (E)-7-[4-(4-FLUOROPHENYL)-6-ISOPROPYL-2-[METHYL(METHYLSULFONYL)AMINO] PYRIMIDIN-5-YL](3R,5S)-3,5-DIHYDROXYHEPT-6-ENOIC ACID AND CRYSTALLINE INTERMEDIATES THEREOF
EN - PROCESS FOR THE MANUFACTURE OF THE CALCIUM SALT OF ROSUVASTATIN (E)-7-[4-(4-FLUOROPHENYL)-6-ISOPROPYL-2-[METHYL(METHYLSULFONYL)AMINO] PYRIMIDIN-5-YL](3R,5S)-3,5-DIHYDROXYHEPT-6-ENOIC ACID AND CRYSTALLINE INTERMEDIATES THEREOF

Teisinis statusas

Patentas neįsigaliojo (pagal Susitarimą)

Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) INT.CL. C07D 405/06
C07D 239/42
Europos patentas
(11) Patento numeris 1682536
(13) Dokumento rūšis T
(96) Europos patento paraiškos numeris 04768997.1
Europos patento paraiškos padavimo data 2004-10-22
(97) Europos patento paraiškos paskelbimo data 2006-07-26
(45) Paskelbimo apie Europos patento išdavimą data 2013-02-27
(46) Apibrėžties vertimo paskelbimo data
Tarptautinės paraiškos padavimo
(86) Numeris PCT/GB2004/004481
Data 2004-10-22
Tarptautinės paraiškos paskelbimo
(87) Numeris WO 2005/042522
Data 2005-05-12
Prioriteto paraiškos
(30) Numeris Data Šalis
0324791 2003-10-24 GB
Išradėjai
(72)
OKADA, Tetsuo, Shionogi & Company Limited, JP
HORBURY, John, AstraZeneca, GB
LAFFAN, David Dermot Patrick, AstraZeneca, GB
Savininkas
(73) AstraZeneca UK Limited, 2 Kingdom Street, London W2 6BD, GB
SHIONOGI & CO., LTD., 1-8, Doshomachi 3-chome, Chuo-ku, Osaka 541-0045, JP
Pavadinimas
(54) PROCESS FOR THE MANUFACTURE OF THE CALCIUM SALT OF ROSUVASTATIN (E)-7-[4-(4-FLUOROPHENYL)-6-ISOPROPYL-2-[METHYL(METHYLSULFONYL)AMINO] PYRIMIDIN-5-YL](3R,5S)-3,5-DIHYDROXYHEPT-6-ENOIC ACID AND CRYSTALLINE INTERMEDIATES THEREOF
  PROCESS FOR THE MANUFACTURE OF THE CALCIUM SALT OF ROSUVASTATIN (E)-7-[4-(4-FLUOROPHENYL)-6-ISOPROPYL-2-[METHYL(METHYLSULFONYL)AMINO] PYRIMIDIN-5-YL](3R,5S)-3,5-DIHYDROXYHEPT-6-ENOIC ACID AND CRYSTALLINE INTERMEDIATES THEREOF