Herbas VPB

Print
EN | LT
LT - GALACTOSYLATED PRO-DRUGS OF NON-STEROIDAL ANTI-INFLAMMATORIES WITH IMPROVED PHARMACOKINETIC CHARACTERISTICS AND REDUCED TOXICITY OF THE STARTING DRUG
EN - GALACTOSYLATED PRO-DRUGS OF NON-STEROIDAL ANTI-INFLAMMATORIES WITH IMPROVED PHARMACOKINETIC CHARACTERISTICS AND REDUCED TOXICITY OF THE STARTING DRUG

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. A61K 47/48
A61P 29/00
C07H 13/02
C07H 13/04
C07H 13/08
C07H 13/10
A61K 31/7024
European patent
(11) Number of the document 2320951
(13) Kind of document T
(96) European patent application number 09787810.2
Date of filing the European patent application 2009-07-29
(97) Date of publication of the European application 2011-05-18
(45) Date of publication and mention of the grant of the patent 2016-01-06
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/IT2009/000341
Date 2009-07-29
PCT application publication
(87) Number WO 2010/013279
Date 2010-02-04
Priority applications
(30) Number Date Country code
NA20080047 2008-07-29 IT
Inventors
(72)
ABIGNENTE, Enrico, IT
MELISI, Daniela, IT
CURCIO, Annalisa, IT
LUONGO, Elvira, IT
LA RANA, Giovanna, IT
SASSO, Oscar, IT
SARNELLI, Giovanni, IT
RUSSO, Roberto, IT
NIEDDU, Maria, IT
CIRILLO, Carla, IT
DE LUCIA, Salvatore, IT
Grantee
(73) Calignano, Antonio, Corso Amedeo di Savoia 239, 801369 Napoli Na, IT
Stewart Italia SRL, Corso G. Matteotti 10, 20121 Milano, IT
Rimoli, Maria Grazia, Via San Nullo 64, 80014 Giugliano (NA), IT
Cuomo, Rosario, Via Martiri delle Foibe 11, 81100 Caserta, IT
Boatto, Gianpiero, Via delle Magnolie 43/B, 07100 Sassari, IT
Title
(54) GALACTOSYLATED PRO-DRUGS OF NON-STEROIDAL ANTI-INFLAMMATORIES WITH IMPROVED PHARMACOKINETIC CHARACTERISTICS AND REDUCED TOXICITY OF THE STARTING DRUG
  GALACTOSYLATED PRO-DRUGS OF NON-STEROIDAL ANTI-INFLAMMATORIES WITH IMPROVED PHARMACOKINETIC CHARACTERISTICS AND REDUCED TOXICITY OF THE STARTING DRUG