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Legal status
Patent not validated
(51) | INT.CL. | A61K 47/48 | |
A61P 29/00 | |||
C07H 13/02 | |||
C07H 13/04 | |||
C07H 13/08 | |||
C07H 13/10 | |||
A61K 31/7024 |
(11) | Number of the document | 2320951 |
(13) | Kind of document | T |
(96) | European patent application number | 09787810.2 |
Date of filing the European patent application | 2009-07-29 | |
(97) | Date of publication of the European application | 2011-05-18 |
(45) | Date of publication and mention of the grant of the patent | 2016-01-06 |
(46) | Date of publication of the claims translation |
(86) | Number | PCT/IT2009/000341 |
Date | 2009-07-29 |
(87) | Number | WO 2010/013279 |
Date | 2010-02-04 |
(30) | Number | Date | Country code |
NA20080047 | 2008-07-29 | IT |
(72) |
ABIGNENTE, Enrico, IT
MELISI, Daniela, IT
CURCIO, Annalisa, IT
LUONGO, Elvira, IT
LA RANA, Giovanna, IT
SASSO, Oscar, IT
SARNELLI, Giovanni, IT
RUSSO, Roberto, IT
NIEDDU, Maria, IT
CIRILLO, Carla, IT
DE LUCIA, Salvatore, IT
|
(73) |
Calignano, Antonio,
Corso Amedeo di Savoia 239, 801369 Napoli Na,
IT
Stewart Italia SRL, Corso G. Matteotti 10, 20121 Milano, IT Rimoli, Maria Grazia, Via San Nullo 64, 80014 Giugliano (NA), IT Cuomo, Rosario, Via Martiri delle Foibe 11, 81100 Caserta, IT Boatto, Gianpiero, Via delle Magnolie 43/B, 07100 Sassari, IT |
(54) | GALACTOSYLATED PRO-DRUGS OF NON-STEROIDAL ANTI-INFLAMMATORIES WITH IMPROVED PHARMACOKINETIC CHARACTERISTICS AND REDUCED TOXICITY OF THE STARTING DRUG |
GALACTOSYLATED PRO-DRUGS OF NON-STEROIDAL ANTI-INFLAMMATORIES WITH IMPROVED PHARMACOKINETIC CHARACTERISTICS AND REDUCED TOXICITY OF THE STARTING DRUG |