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LT - GALACTOSYLATED PRO-DRUGS OF NON-STEROIDAL ANTI-INFLAMMATORIES WITH IMPROVED PHARMACOKINETIC CHARACTERISTICS AND REDUCED TOXICITY OF THE STARTING DRUG
EN - GALACTOSYLATED PRO-DRUGS OF NON-STEROIDAL ANTI-INFLAMMATORIES WITH IMPROVED PHARMACOKINETIC CHARACTERISTICS AND REDUCED TOXICITY OF THE STARTING DRUG

Teisinis statusas

Patentas neįsigaliojo (pagal EPK)

Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) INT.CL. A61K 47/48
A61P 29/00
C07H 13/02
C07H 13/04
C07H 13/08
C07H 13/10
A61K 31/7024
Europos patentas
(11) Patento numeris 2320951
(13) Dokumento rūšis T
(96) Europos patento paraiškos numeris 09787810.2
Europos patento paraiškos padavimo data 2009-07-29
(97) Europos patento paraiškos paskelbimo data 2011-05-18
(45) Paskelbimo apie Europos patento išdavimą data 2016-01-06
(46) Apibrėžties vertimo paskelbimo data
Tarptautinės paraiškos padavimo
(86) Numeris PCT/IT2009/000341
Data 2009-07-29
Tarptautinės paraiškos paskelbimo
(87) Numeris WO 2010/013279
Data 2010-02-04
Prioriteto paraiškos
(30) Numeris Data Šalis
NA20080047 2008-07-29 IT
Išradėjai
(72)
ABIGNENTE, Enrico, IT
MELISI, Daniela, IT
CURCIO, Annalisa, IT
LUONGO, Elvira, IT
LA RANA, Giovanna, IT
SASSO, Oscar, IT
SARNELLI, Giovanni, IT
RUSSO, Roberto, IT
NIEDDU, Maria, IT
CIRILLO, Carla, IT
DE LUCIA, Salvatore, IT
Savininkas
(73) Calignano, Antonio, Corso Amedeo di Savoia 239, 801369 Napoli Na, IT
Stewart Italia SRL, Corso G. Matteotti 10, 20121 Milano, IT
Rimoli, Maria Grazia, Via San Nullo 64, 80014 Giugliano (NA), IT
Cuomo, Rosario, Via Martiri delle Foibe 11, 81100 Caserta, IT
Boatto, Gianpiero, Via delle Magnolie 43/B, 07100 Sassari, IT
Pavadinimas
(54) GALACTOSYLATED PRO-DRUGS OF NON-STEROIDAL ANTI-INFLAMMATORIES WITH IMPROVED PHARMACOKINETIC CHARACTERISTICS AND REDUCED TOXICITY OF THE STARTING DRUG
  GALACTOSYLATED PRO-DRUGS OF NON-STEROIDAL ANTI-INFLAMMATORIES WITH IMPROVED PHARMACOKINETIC CHARACTERISTICS AND REDUCED TOXICITY OF THE STARTING DRUG