![]() |
![]() |
Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
(51) | INT.CL. | C07D 405/12 | |
A61K 31/404 | |||
A61P 11/00 |
(11) | Patento numeris | 2563778 |
(13) | Dokumento rūšis | T |
(96) | Europos patento paraiškos numeris | 11713134.2 |
Europos patento paraiškos padavimo data | 2011-03-25 | |
(97) | Europos patento paraiškos paskelbimo data | 2013-03-06 |
(45) | Paskelbimo apie Europos patento išdavimą data | 2016-08-24 |
(46) | Apibrėžties vertimo paskelbimo data |
(86) | Numeris | PCT/US2011/030032 |
Data | 2011-03-25 |
(87) | Numeris | WO 2011/119984 |
Data | 2011-09-29 |
(30) | Numeris | Data | Šalis |
321636 P | 2010-04-07 | US | |
321561 P | 2010-04-07 | US | |
319953 P | 2010-04-01 | US | |
317376 P | 2010-03-25 | US |
(72) |
KESHAVARZ-SHOKRI, Ali, US
ZHANG, Beili, US
ALCACIO, Tim, Edward, US
LEE, Elaine, Chungmin, US
ZHANG, Yuegang, US
KRAWIEC, Mariusz, US
|
(73) |
Vertex Pharmaceuticals Incorporated,
50 Northern Avenue, Boston, MA 02210,
US
|
(54) | CRYSTALLINE FORM OF (R)-1(2,2 -DIFLUOROBENZO[D][1,3]DIOXOL-5YL)-N-(1-(2,3-DIHYDEROXYPROPYL)-6-FLUORO-2-(1-HYDROXY-2-METHYLPROPAN-2YL)-1H-INDOL-5YL)CYCLOPROPANECARBOXAMIDE |
CRYSTALLINE FORM OF (R)-1(2,2 -DIFLUOROBENZO[D][1,3]DIOXOL-5YL)-N-(1-(2,3-DIHYDEROXYPROPYL)-6-FLUORO-2-(1-HYDROXY-2-METHYLPROPAN-2YL)-1H-INDOL-5YL)CYCLOPROPANECARBOXAMIDE |