Herbas VPB

Print
EN | LT
LT - N-[5-(AMINOSULFONYL)-4-METHYL-1,3-THIAZOL-2-YL]-N-METHYL-2-[4-(2-PYRIDINYL)PHENYL]ACETAMIDE MESYLATE MONOHYDRATE HAVING A SPECIFIC PARTICLE SIZE DISTRIBUTION RANGE AND A SPECIFIC SURFACE AREA RANGE FOR USE IN PHARMACEUTICAL FORMULATIONS.
EN - N-[5-(AMINOSULFONYL)-4-METHYL-1,3-THIAZOL-2-YL]-N-METHYL-2-[4-(2-PYRIDINYL)PHENYL]ACETAMIDE MESYLATE MONOHYDRATE HAVING A SPECIFIC PARTICLE SIZE DISTRIBUTION RANGE AND A SPECIFIC SURFACE AREA RANGE FOR USE IN PHARMACEUTICAL FORMULATIONS.

Legal status

Patent not validated

Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07D 417/12
A61K 31/4402
A61P 31/00
A61P 31/22
European patent
(11) Number of the document 2598502
(13) Kind of document T
(96) European patent application number 12762305.6
Date of filing the European patent application 2012-09-26
(97) Date of publication of the European application 2013-06-05
(45) Date of publication and mention of the grant of the patent 2014-05-14
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/EP2012/068958
Date 2012-09-26
PCT application publication
(87) Number WO 2013/045491
Date 2013-04-04
Priority applications
(30) Number Date Country code
PCT/EP2011/0078 2011-09-26 WO
Inventors
(72)
Schwab, Wilfried, DE
Birkmann, Alexander, DE
Paulus, Kerstin, DE
Vögtli, Kurt, DE
Haag, Dieter, DE
Mass, Stephan, DE
Ruepp, Kristian, DE
Grantee
(73) AiCuris GmbH & Co. KG, Friedrich-Ebert-Strasse 475, 42117 Wuppertal, DE
Title
(54) N-[5-(AMINOSULFONYL)-4-METHYL-1,3-THIAZOL-2-YL]-N-METHYL-2-[4-(2-PYRIDINYL)PHENYL]ACETAMIDE MESYLATE MONOHYDRATE HAVING A SPECIFIC PARTICLE SIZE DISTRIBUTION RANGE AND A SPECIFIC SURFACE AREA RANGE FOR USE IN PHARMACEUTICAL FORMULATIONS.
  N-[5-(AMINOSULFONYL)-4-METHYL-1,3-THIAZOL-2-YL]-N-METHYL-2-[4-(2-PYRIDINYL)PHENYL]ACETAMIDE MESYLATE MONOHYDRATE HAVING A SPECIFIC PARTICLE SIZE DISTRIBUTION RANGE AND A SPECIFIC SURFACE AREA RANGE FOR USE IN PHARMACEUTICAL FORMULATIONS.