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Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
(51) | INT.CL. | C07D 417/12 | |
A61K 31/4402 | |||
A61P 31/00 | |||
A61P 31/22 |
(11) | Patento numeris | 2598502 |
(13) | Dokumento rūšis | T |
(96) | Europos patento paraiškos numeris | 12762305.6 |
Europos patento paraiškos padavimo data | 2012-09-26 | |
(97) | Europos patento paraiškos paskelbimo data | 2013-06-05 |
(45) | Paskelbimo apie Europos patento išdavimą data | 2014-05-14 |
(46) | Apibrėžties vertimo paskelbimo data |
(86) | Numeris | PCT/EP2012/068958 |
Data | 2012-09-26 |
(87) | Numeris | WO 2013/045491 |
Data | 2013-04-04 |
(30) | Numeris | Data | Šalis |
PCT/EP2011/0078 | 2011-09-26 | WO |
(72) |
Schwab, Wilfried, DE
Birkmann, Alexander, DE
Paulus, Kerstin, DE
Vögtli, Kurt, DE
Haag, Dieter, DE
Mass, Stephan, DE
Ruepp, Kristian, DE
|
(73) |
AiCuris GmbH & Co. KG,
Friedrich-Ebert-Strasse 475, 42117 Wuppertal,
DE
|
(54) | N-[5-(AMINOSULFONYL)-4-METHYL-1,3-THIAZOL-2-YL]-N-METHYL-2-[4-(2-PYRIDINYL)PHENYL]ACETAMIDE MESYLATE MONOHYDRATE HAVING A SPECIFIC PARTICLE SIZE DISTRIBUTION RANGE AND A SPECIFIC SURFACE AREA RANGE FOR USE IN PHARMACEUTICAL FORMULATIONS. |
N-[5-(AMINOSULFONYL)-4-METHYL-1,3-THIAZOL-2-YL]-N-METHYL-2-[4-(2-PYRIDINYL)PHENYL]ACETAMIDE MESYLATE MONOHYDRATE HAVING A SPECIFIC PARTICLE SIZE DISTRIBUTION RANGE AND A SPECIFIC SURFACE AREA RANGE FOR USE IN PHARMACEUTICAL FORMULATIONS. |