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EN | LT
LT - Use of (S)-pyrrolidine-1,2-dicarboxylic acid 2-amide 1-({4-methyl-5-[2-(2,2,2-trifluoro-1,1-dimethyl-ethyl)- pyridin-4-yl]-thiazol-2-yl}-amide) in the treatment of EGFR dependent diseases or diseases that have acquired resistance to agents that target E
EN - Use of (S)-pyrrolidine-1,2-dicarboxylic acid 2-amide 1-({4-methyl-5-[2-(2,2,2-trifluoro-1,1-dimethyl-ethyl)- pyridin-4-yl]-thiazol-2-yl}-amide) in the treatment of EGFR dependent diseases or diseases that have acquired resistance to agents that target E

Teisinis statusas

Patentas neįsigaliojo (pagal EPK)

Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) INT.CL. A61K 31/4439
A61K 31/517
A61K 39/395
A61K 45/06
A61P 35/00
C07K 16/32
A61K 39/00
Europos patentas
(11) Patento numeris 2637661
(13) Dokumento rūšis T
(96) Europos patento paraiškos numeris 11782111.6
Europos patento paraiškos padavimo data 2011-11-07
(97) Europos patento paraiškos paskelbimo data 2013-09-18
(45) Paskelbimo apie Europos patento išdavimą data 2017-12-20
(46) Apibrėžties vertimo paskelbimo data
Tarptautinės paraiškos padavimo
(86) Numeris PCT/EP2011/069522
Data 2011-11-07
Tarptautinės paraiškos paskelbimo
(87) Numeris WO 2012/062694
Data 2012-05-18
Prioriteto paraiškos
(30) Numeris Data Šalis
411117 P 2010-11-08 US
Išradėjai
(72)
BRACHMANN, Saskia Maria, CH
FRITSCH, Christine, CH
MAIRA, Sauveur-Michel, CH
SCHNELL, Christian René, CH
GARCIA-ECHEVERRIA, Carlos, FR
Savininkas
(73) Novartis AG, Lichtstrasse 35, 4056 Basel, CH
Pavadinimas
(54) Use of (S)-pyrrolidine-1,2-dicarboxylic acid 2-amide 1-({4-methyl-5-[2-(2,2,2-trifluoro-1,1-dimethyl-ethyl)- pyridin-4-yl]-thiazol-2-yl}-amide) in the treatment of EGFR dependent diseases or diseases that have acquired resistance to agents that target E
  Use of (S)-pyrrolidine-1,2-dicarboxylic acid 2-amide 1-({4-methyl-5-[2-(2,2,2-trifluoro-1,1-dimethyl-ethyl)- pyridin-4-yl]-thiazol-2-yl}-amide) in the treatment of EGFR dependent diseases or diseases that have acquired resistance to agents that target E