LT - PHARMACEUTICALLY ACCEPTABLE SALT OF (E)-N-[4-[[3-CHLORO-4-(2-PYRIDYLMETHOXY)PHENYL]AMINO]-3-CYANO-7-ETHOXY-6-QUINOLYL]-3-[(2R)-1-METHYLPYRROLIDIN-2-YL]PROP-2-ENAMIDE, PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF
EN - PHARMACEUTICALLY ACCEPTABLE SALT OF (E)-N-[4-[[3-CHLORO-4-(2-PYRIDYLMETHOXY)PHENYL]AMINO]-3-CYANO-7-ETHOXY-6-QUINOLYL]-3-[(2R)-1-METHYLPYRROLIDIN-2-YL]PROP-2-ENAMIDE, PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF
Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) |
INT.CL. |
C07D 401/14 |
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A61K 31/4709 |
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A61P 35/00 |
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Europos patentas
(11) |
Patento numeris |
2684877 |
(13) |
Dokumento rūšis |
T |
(96) |
Europos patento paraiškos numeris |
12757831.8 |
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Europos patento paraiškos padavimo data |
2012-02-10 |
(97) |
Europos patento paraiškos paskelbimo data |
2014-01-15 |
(45) |
Paskelbimo apie Europos patento išdavimą data |
2016-10-19
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(46) |
Apibrėžties vertimo paskelbimo data |
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Tarptautinės paraiškos padavimo
(86) |
Numeris |
PCT/CN2012/071015 |
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Data |
2012-02-10 |
Tarptautinės paraiškos paskelbimo
(87) |
Numeris |
WO 2012/122865 |
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Data |
2012-09-20 |
Prioriteto paraiškos
(30) |
Numeris |
Data |
Šalis |
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201110062359 |
2011-03-11
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CN |
Išradėjai
(72) |
LI, Xin, CN
WANG, Bin, CN
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Savininkas
(73) |
Shanghai Hengrui Pharmaceutical Co. Ltd.,
279 Wenjing Road, Minhang District Shanghai 200245,
CN
Jiangsu Hengrui Medicine Co. Ltd.,
No. 7 Kunlunshan Road Economic and Technological Development Zone Lianyungang, Jiangsu 222047,
CN
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Pavadinimas
(54) |
PHARMACEUTICALLY ACCEPTABLE SALT OF (E)-N-[4-[[3-CHLORO-4-(2-PYRIDYLMETHOXY)PHENYL]AMINO]-3-CYANO-7-ETHOXY-6-QUINOLYL]-3-[(2R)-1-METHYLPYRROLIDIN-2-YL]PROP-2-ENAMIDE, PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF |
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PHARMACEUTICALLY ACCEPTABLE SALT OF (E)-N-[4-[[3-CHLORO-4-(2-PYRIDYLMETHOXY)PHENYL]AMINO]-3-CYANO-7-ETHOXY-6-QUINOLYL]-3-[(2R)-1-METHYLPYRROLIDIN-2-YL]PROP-2-ENAMIDE, PREPARATION METHOD THEREFOR, AND MEDICAL USE THEREOF |