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LT - PROCESS FOR THE PREPARATION OF (R)-3-(6-(4-METHYLPHENYL)-PYRIDIN-3-YLOXY)-1-AZA-BICYCLO[2.2.2]OCTANE BY REACTING 5-CHLORO-2-(4-METHYLPHENYL)PYRIDINE WITH (R)-3-HYDROXY-1-AZA-BICYCLO[2.2.2]OCTANE
EN - PROCESS FOR THE PREPARATION OF (R)-3-(6-(4-METHYLPHENYL)-PYRIDIN-3-YLOXY)-1-AZA-BICYCLO[2.2.2]OCTANE BY REACTING 5-CHLORO-2-(4-METHYLPHENYL)PYRIDINE WITH (R)-3-HYDROXY-1-AZA-BICYCLO[2.2.2]OCTANE

Teisinis statusas

Patentas neįsigaliojo (pagal EPK)

Bibliografiniai duomenys
Tarptautinės patentų klasifikacijos indeksai (TPK)
(51) INT.CL. C07D 453/02
A61K 31/439
A61P 25/16
A61P 25/18
A61P 25/22
A61P 25/24
A61P 25/28
Europos patentas
(11) Patento numeris 3075732
(13) Dokumento rūšis T
(96) Europos patento paraiškos numeris 16162555.3
Europos patento paraiškos padavimo data 2012-07-12
(97) Europos patento paraiškos paskelbimo data 2016-10-05
(45) Paskelbimo apie Europos patento išdavimą data 2018-09-12
(46) Apibrėžties vertimo paskelbimo data
Prioriteto paraiškos
(30) Numeris Data Šalis
201161508147 P 2011-07-15 US
Išradėjai
(72)
MARTERER, Wolfgang, CH
PRASHAD, Mahavir, US
VILLHAUER, Edwin Bernard, US
WAYKOLE, Liladhar Murlidhar, US
VIVELO, James Anthony, US
SUTTER, Bertrand, CH
BIANCHI, Jean-Claude, CH
WU, Raeann, US
HAR, Denis, US
KARPINSKI, Piotr H., US
PIGNONE, Massimo, CH
STINGELIN, Doris, CH
BUERGER, Eckart, CH
Savininkas
(73) Novartis AG, Lichtstrasse 35, 4056 Basel, CH
Pavadinimas
(54) PROCESS FOR THE PREPARATION OF (R)-3-(6-(4-METHYLPHENYL)-PYRIDIN-3-YLOXY)-1-AZA-BICYCLO[2.2.2]OCTANE BY REACTING 5-CHLORO-2-(4-METHYLPHENYL)PYRIDINE WITH (R)-3-HYDROXY-1-AZA-BICYCLO[2.2.2]OCTANE
  PROCESS FOR THE PREPARATION OF (R)-3-(6-(4-METHYLPHENYL)-PYRIDIN-3-YLOXY)-1-AZA-BICYCLO[2.2.2]OCTANE BY REACTING 5-CHLORO-2-(4-METHYLPHENYL)PYRIDINE WITH (R)-3-HYDROXY-1-AZA-BICYCLO[2.2.2]OCTANE