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Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
| (51) | INT.CL. | C07D 453/02 | |
| A61K 31/439 | |||
| A61P 25/16 | |||
| A61P 25/18 | |||
| A61P 25/22 | |||
| A61P 25/24 | |||
| A61P 25/28 |
| (11) | Patento numeris | 3075732 |
| (13) | Dokumento rūšis | T |
| (96) | Europos patento paraiškos numeris | 16162555.3 |
| Europos patento paraiškos padavimo data | 2012-07-12 | |
| (97) | Europos patento paraiškos paskelbimo data | 2016-10-05 |
| (45) | Paskelbimo apie Europos patento išdavimą data | 2018-09-12 |
| (46) | Apibrėžties vertimo paskelbimo data |
| (30) | Numeris | Data | Šalis |
| 201161508147 P | 2011-07-15 | US |
| (72) |
MARTERER, Wolfgang, CH
PRASHAD, Mahavir, US
VILLHAUER, Edwin Bernard, US
WAYKOLE, Liladhar Murlidhar, US
VIVELO, James Anthony, US
SUTTER, Bertrand, CH
BIANCHI, Jean-Claude, CH
WU, Raeann, US
HAR, Denis, US
KARPINSKI, Piotr H., US
PIGNONE, Massimo, CH
STINGELIN, Doris, CH
BUERGER, Eckart, CH
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| (73) |
Novartis AG,
Lichtstrasse 35, 4056 Basel,
CH
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| (54) | PROCESS FOR THE PREPARATION OF (R)-3-(6-(4-METHYLPHENYL)-PYRIDIN-3-YLOXY)-1-AZA-BICYCLO[2.2.2]OCTANE BY REACTING 5-CHLORO-2-(4-METHYLPHENYL)PYRIDINE WITH (R)-3-HYDROXY-1-AZA-BICYCLO[2.2.2]OCTANE |
| PROCESS FOR THE PREPARATION OF (R)-3-(6-(4-METHYLPHENYL)-PYRIDIN-3-YLOXY)-1-AZA-BICYCLO[2.2.2]OCTANE BY REACTING 5-CHLORO-2-(4-METHYLPHENYL)PYRIDINE WITH (R)-3-HYDROXY-1-AZA-BICYCLO[2.2.2]OCTANE |