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LT - PROCESS FOR THE PREPARATION OF TERT-BUTYL 4-((2S,5R)-6-(BENZYLOXY)-7-OXO-1,6-DIAZABICYCLO[3.2.1]OCTANE-2-CARBOXAMIDO)PIPERIDINE-1-CARBOXYLATE AND ANALOGS THEREOF
EN - PROCESS FOR THE PREPARATION OF TERT-BUTYL 4-((2S,5R)-6-(BENZYLOXY)-7-OXO-1,6-DIAZABICYCLO[3.2.1]OCTANE-2-CARBOXAMIDO)PIPERIDINE-1-CARBOXYLATE AND ANALOGS THEREOF

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Bibliographic data
Indications of the International Patent Classification (IPC)
(51) INT.CL. C07F 7/10
C07F 7/18
C07D 471/08
European patent
(11) Number of the document 3227306
(13) Kind of document T
(96) European patent application number 15865871.6
Date of filing the European patent application 2015-11-30
(97) Date of publication of the European application 2017-10-11
(45) Date of publication and mention of the grant of the patent 2020-07-15
(46) Date of publication of the claims translation
PCT application
(86) Number PCT/US2015/062884
Date 2015-11-30
PCT application publication
(87) Number WO 2016/089718
Date 2016-06-09
Priority applications
(30) Number Date Country code
201462086420 P 2014-12-02 US
Inventors
(72)
LIU, Zhijian, US
YASUDA, Nobuyoshi, US
YANG, Lu, US
KLAPARS, Artis, US
CAMPOS, Kevin R., US
REIBARKH, Mikhail, US
Grantee
(73) Merck Sharp & Dohme Corp., 126 East Lincoln Avenue, Rahway, NJ 07065-0907, US
Title
(54) PROCESS FOR THE PREPARATION OF TERT-BUTYL 4-((2S,5R)-6-(BENZYLOXY)-7-OXO-1,6-DIAZABICYCLO[3.2.1]OCTANE-2-CARBOXAMIDO)PIPERIDINE-1-CARBOXYLATE AND ANALOGS THEREOF
  PROCESS FOR THE PREPARATION OF TERT-BUTYL 4-((2S,5R)-6-(BENZYLOXY)-7-OXO-1,6-DIAZABICYCLO[3.2.1]OCTANE-2-CARBOXAMIDO)PIPERIDINE-1-CARBOXYLATE AND ANALOGS THEREOF