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Teisinis statusas
Patentas neįsigaliojo (pagal EPK)
(51) | INT.CL. | C07F 7/10 | |
C07F 7/18 | |||
C07D 471/08 |
(11) | Patento numeris | 3227306 |
(13) | Dokumento rūšis | T |
(96) | Europos patento paraiškos numeris | 15865871.6 |
Europos patento paraiškos padavimo data | 2015-11-30 | |
(97) | Europos patento paraiškos paskelbimo data | 2017-10-11 |
(45) | Paskelbimo apie Europos patento išdavimą data | 2020-07-15 |
(46) | Apibrėžties vertimo paskelbimo data |
(86) | Numeris | PCT/US2015/062884 |
Data | 2015-11-30 |
(87) | Numeris | WO 2016/089718 |
Data | 2016-06-09 |
(30) | Numeris | Data | Šalis |
201462086420 P | 2014-12-02 | US |
(72) |
LIU, Zhijian, US
YASUDA, Nobuyoshi, US
YANG, Lu, US
KLAPARS, Artis, US
CAMPOS, Kevin R., US
REIBARKH, Mikhail, US
|
(73) |
Merck Sharp & Dohme Corp.,
126 East Lincoln Avenue, Rahway, NJ 07065-0907,
US
|
(54) | PROCESS FOR THE PREPARATION OF TERT-BUTYL 4-((2S,5R)-6-(BENZYLOXY)-7-OXO-1,6-DIAZABICYCLO[3.2.1]OCTANE-2-CARBOXAMIDO)PIPERIDINE-1-CARBOXYLATE AND ANALOGS THEREOF |
PROCESS FOR THE PREPARATION OF TERT-BUTYL 4-((2S,5R)-6-(BENZYLOXY)-7-OXO-1,6-DIAZABICYCLO[3.2.1]OCTANE-2-CARBOXAMIDO)PIPERIDINE-1-CARBOXYLATE AND ANALOGS THEREOF |